SCHEMBL24326765

SCHEMBL24326765

CNc1nc(O)cc(-c2c(C)cccc2C)n1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.43
NUDT1 P36639 5/20 0.37
HSD17B10 Q99714 1/20 0.36
HSP90AA1 P07900 1/20 0.34
HTR7 P34969 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
IDH2 P48735 1/20 0.33
ALDH1A1 P00352 1/20 0.33
PLK1 P53350 1/20 0.33
TLR8 Q9NR97 1/20 0.33
GAA P10253 1/20 0.33
SRC P12931 1/20 0.32
GPR39 O43194 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24326363 0.83 TDP1 (0.46) TDP1NUDT1HSP90AA1HTR7IDH2
SCHEMBL24329987 0.79 PLK1 (0.35) NUDT1PLK1
SCHEMBL24331435 0.77 HSP90AA1 (0.50) TDP1NUDT1HSP90AA1HTR7ADORA2A
SCHEMBL10429480 0.73 TDP1 (0.41) TDP1NUDT1HSD17B10ADORA2AADORA1
SCHEMBL24298907 0.72 PARP1 (0.38)
SCHEMBL24299252 0.72 CYP1A2 (0.40) TDP1HSD17B10SRC
SCHEMBL10285741 0.70 MAPT (0.46) TDP1HSD17B10ALDH1A1GAA
SCHEMBL12658527 0.69 TDP1 (0.35) TDP1HSD17B10ADORA2AADORA1IDH2
SCHEMBL20008234 0.64 CYP1A2 (0.49) TDP1NUDT1HSD17B10HSP90AA1ALDH1A1
SCHEMBL26354524 0.63 NOS2 (0.45) TDP1HSP90AA1HTR7ALDH1A1TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022076625-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed