SCHEMBL24327370

SCHEMBL24327370

Cn1cc(-c2nc(-c3ccc(Cl)cc3)cnc2CN)cn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR3 P22607 3/20 0.51
KDR P35968 1/20 0.51
CSF1R P07333 3/20 0.46
KCNH2 Q12809 1/20 0.43
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42
FLT3 P36888 2/20 0.41
LOXL2 Q9Y4K0 1/20 0.41
MAPK1 P28482 3/20 0.40
AURKA O14965 1/20 0.40
AURKB Q96GD4 1/20 0.40
FGFR1 P11362 2/20 0.40
FGFR2 P21802 2/20 0.40
FGFR4 P22455 1/20 0.40
CHEK1 O14757 1/20 0.40
PRMT5 O14744 2/20 0.39
WDR77 Q9BQA1 2/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24327347 0.90 KDR (0.53) FGFR3KDRCSF1RKCNH2CNR1
SCHEMBL29498933 0.90 KDR (0.53) FGFR3KDRCSF1RKCNH2CNR1
SCHEMBL24328703 0.87 FGFR3 (0.51) FGFR3KDRCSF1RKCNH2CNR1
SCHEMBL24327827 0.84 FGFR3 (0.53) FGFR3KDRCSF1RMAPK1AURKA
SCHEMBL29498949 0.84 FGFR3 (0.56) FGFR3KDRCSF1RKCNH2CNR1
SCHEMBL24327350 0.84 FGFR3 (0.56) FGFR3KDRCSF1RKCNH2CNR1
SCHEMBL24327324 0.81 FGFR3 (0.50) FGFR3KDRCSF1RKCNH2CNR1
SCHEMBL24328713 0.80 CNR1 (0.52) FGFR3KDRKCNH2CNR1CNR2
SCHEMBL28724019 0.80 FGFR3 (0.51) FGFR3KDRCSF1RKCNH2CNR1
SCHEMBL24327348 0.79 CHRM1 (0.46) FGFR3KDRCSF1RKCNH2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114369097-B Heteroaromatic AhR inhibitors 山东轩竹医药科技有限公司 2023-07-14 CN disclosed
WO-2022078356-A1 HETEROAROMATIC AHR INHIBITOR 山东轩竹医药科技有限公司 2022-04-21 WO disclosed
WO-2022078356-A1 HETEROAROMATIC AHR INHIBITOR 山东轩竹医药科技有限公司 2022-04-21 WO disclosed
CN-114369097-A Heteroaromatic AhR inhibitors 山东轩竹医药科技有限公司 2022-04-19 CN disclosed