SCHEMBL24328703

SCHEMBL24328703

Cn1cc(-c2nc(-c3ccc(Cl)cc3)cnc2CO)cn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR3 P22607 5/20 0.51
KDR P35968 3/20 0.51
CNR1 P21554 1/20 0.44
CNR2 P34972 1/20 0.44
KCNH2 Q12809 1/20 0.43
CHEK1 O14757 1/20 0.42
FGFR1 P11362 4/20 0.42
FGFR2 P21802 4/20 0.42
FGFR4 P22455 3/20 0.42
FLT3 P36888 4/20 0.41
CSF1R P07333 3/20 0.41
MAPK1 P28482 3/20 0.40
AURKA O14965 1/20 0.40
AURKB Q96GD4 1/20 0.40
CLK1 P49759 1/20 0.40
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
TYK2 P29597 1/20 0.39
JAK3 P52333 1/20 0.39
MET P08581 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24327347 0.90 KDR (0.53) FGFR3KDRCNR1CNR2KCNH2
SCHEMBL29498933 0.90 KDR (0.53) FGFR3KDRCNR1CNR2KCNH2
SCHEMBL24327370 0.87 FGFR3 (0.51) FGFR3KDRCNR1CNR2KCNH2
SCHEMBL24327350 0.84 FGFR3 (0.56) FGFR3KDRCNR1CNR2KCNH2
SCHEMBL29498949 0.84 FGFR3 (0.56) FGFR3KDRCNR1CNR2KCNH2
SCHEMBL24327827 0.82 FGFR3 (0.53) FGFR3KDRFGFR1FGFR2CSF1R
SCHEMBL24328711 0.80 CHEK1 (0.52) FGFR3KDRCNR1CNR2CHEK1
SCHEMBL24328681 0.80 FGFR3 (0.49) FGFR3KDRCNR1CNR2KCNH2
SCHEMBL24328682 0.80 FGFR3 (0.46) FGFR3KDRCHEK1FGFR1FGFR2
SCHEMBL30519232 0.80 FGFR3 (0.46) FGFR3KDRCHEK1FGFR1FGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114369097-B Heteroaromatic AhR inhibitors 山东轩竹医药科技有限公司 2023-07-14 CN disclosed
WO-2022078356-A1 HETEROAROMATIC AHR INHIBITOR 山东轩竹医药科技有限公司 2022-04-21 WO disclosed
WO-2022078356-A1 HETEROAROMATIC AHR INHIBITOR 山东轩竹医药科技有限公司 2022-04-21 WO disclosed
CN-114369097-A Heteroaromatic AhR inhibitors 山东轩竹医药科技有限公司 2022-04-19 CN disclosed