SCHEMBL24327872

SCHEMBL24327872

Cn1cc(-c2nc(-c3ccc(C(F)(F)F)nc3)c[n+](N)c2N)cn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.46
CCNE2 O96020 4/20 0.41
CCNE1 P24864 4/20 0.41
CDK2 P24941 4/20 0.41
CCNB2 O95067 4/20 0.40
CDK1 P06493 4/20 0.40
CCNB1 P14635 4/20 0.40
CDK5 Q00535 4/20 0.40
CDK5R1 Q15078 4/20 0.40
CCNB3 Q8WWL7 4/20 0.40
CCNT1 O60563 3/20 0.40
CDK9 P50750 3/20 0.40
MAP4K4 O95819 1/20 0.38
PIK3CA P42336 1/20 0.38
MINK1 Q8N4C8 1/20 0.38
PI4KB Q9UBF8 1/20 0.38
GRM2 Q14416 1/20 0.38
HSP90AA1 P07900 3/20 0.38
NTRK1 P04629 2/20 0.38
CSF1R P07333 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24327883 0.85 TEK (0.46) KCNH2CDK2FGFR2FGFR3
SCHEMBL24327374 0.82 KCNH2 (0.64) KCNH2CCNE2CCNE1CDK2FGFR2
SCHEMBL29498950 0.82 KCNH2 (0.64) KCNH2CCNE2CCNE1CDK2FGFR2
SCHEMBL29498946 0.82 KCNH2 (0.64) KCNH2CCNE2CCNE1CDK2FGFR2
SCHEMBL24327260 0.80 LRRK2 (0.45) CDK2PIK3CAPI4KBFGFR2FGFR3
SCHEMBL24327354 0.79 CNR1 (0.43) KCNH2CCNE2CCNE1CDK2CCNB2
SCHEMBL24327941 0.79 AXL (0.37) CCNE2CCNE1CDK2CCNB2CDK1
SCHEMBL28724038 0.77 TYK2 (0.39) KCNH2CCNE2CCNE1CDK2CCNB2
SCHEMBL25404864 0.74 MET (0.42) KCNH2MAP4K4GRM2HSP90AA1NTRK1
SCHEMBL28724022 0.72 CCNB2 (0.32) CCNE2CCNE1CDK2CCNB2CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022078356-A1 HETEROAROMATIC AHR INHIBITOR 山东轩竹医药科技有限公司 2022-04-21 WO disclosed