SCHEMBL24328599

SCHEMBL24328599

Clc1nc(N2SN3CCc4cccc2c43)c2cn[nH]c2n1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 2/20 0.35
LMNA P02545 2/20 0.34
MAPT P10636 2/20 0.34
HTT P42858 1/20 0.34
BTK Q06187 1/20 0.33
SGK1 O00141 1/20 0.33
HTR2A P28223 2/20 0.32
HTR2C P28335 2/20 0.32
PAK1 Q13153 2/20 0.31
TRPV1 Q8NER1 2/20 0.31
PDE2A O00408 1/20 0.30
USP2 O75604 1/20 0.30
TP53 P04637 1/20 0.30
GAA P10253 1/20 0.30
ALOX15 P16050 1/20 0.30
MAPK1 P28482 1/20 0.30
BRCA1 P38398 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24351534 0.84 NUDT1 (0.35) RPS6KB1HTR2C
SCHEMBL24327036 0.72 CDK1 (0.39)
SCHEMBL24327019 0.71 ALDH1A1 (0.33) LMNAMAPTMAPK1
SCHEMBL3984786 0.62 PIK3CA (0.49) RPS6KB1LMNAMAPTBTKSGK1
SCHEMBL24328339 0.60 SMN1; SMN2 (0.33)
SCHEMBL55757 0.60 MTOR (0.40) SGK1PDE2A
SCHEMBL560806 0.58 RET (0.52) MAPTHTTBTKHTR2AHTR2C
SCHEMBL24672317 0.58 AKT2 (0.38) BTKSGK1PDE2A
SCHEMBL24327450 0.58 ABL1 (0.31)
SCHEMBL53863 0.58 PLK4 (0.47) LMNABTKPDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022063106-A1 INDOLINE COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS BEIGENE, LTD. (KY) 2022-03-31 WO disclosed