SCHEMBL24328756

SCHEMBL24328756

C[C@@H](C#N)CCc1nnc2c(-c3cnn(C)c3)nc(-c3ccc(Cl)cc3)cn12

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 2/20 0.39
CNR2 P34972 1/20 0.39
JAK2 O60674 8/20 0.34
TYK2 P29597 8/20 0.34
JAK1 P23458 7/20 0.33
JAK3 P52333 3/20 0.33
CYP3A4 P08684 1/20 0.33
KCNH2 Q12809 1/20 0.33
FGFR3 P22607 1/20 0.33
KDR P35968 1/20 0.33
RET P07949 4/20 0.33
CHEK1 O14757 1/20 0.32
CLK1 P49759 1/20 0.32
SCN2A Q99250 1/20 0.32
CECR2 Q9BXF3 1/20 0.32
BAZ2B Q9UIF8 1/20 0.32
BAZ2A Q9UIF9 1/20 0.32
EP300 Q09472 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24328754 0.86 JAK2 (0.39) CNR1CNR2JAK2TYK2JAK1
SCHEMBL24327877 0.82 JAK2 (0.36) CNR1CNR2JAK2TYK2JAK1
SCHEMBL24327880 0.79 CNR1 (0.40) CNR1CNR2JAK2TYK2CYP3A4
SCHEMBL24327876 0.77 CNR1 (0.38) CNR1CNR2JAK2TYK2JAK1
SCHEMBL24327881 0.75 JAK1 (0.37) JAK2TYK2JAK1JAK3CHEK1
SCHEMBL24328759 0.75 TEK (0.41) JAK2TYK2JAK1JAK3KDR
SCHEMBL24327399 0.74 AHR (0.41) CNR1CNR2JAK2TYK2JAK1
SCHEMBL24327391 0.73 JAK2 (0.39) CNR1CNR2JAK2TYK2JAK1
SCHEMBL24327384 0.72 DPP4 (0.32) CYP3A4
SCHEMBL24327848 0.71 JAK2 (0.43) CNR1CNR2JAK2TYK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022078356-A1 HETEROAROMATIC AHR INHIBITOR 山东轩竹医药科技有限公司 2022-04-21 WO disclosed