SCHEMBL24328826

SCHEMBL24328826

C=C(N)N(Cc1ccc(C)cc1)C(=O)Nc1cc(C)cc(C)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
MEN1 O00255 5/20 0.41
KMT2A Q03164 5/20 0.41
POLB P06746 3/20 0.41
GAA P10253 1/20 0.41
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
EGFR P00533 1/20 0.37
ERBB2 P04626 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24327424 0.77 MTOR (0.48) MEN1KMT2APOLBGAASMN1; SMN2
SCHEMBL11142389 0.70 ALDH1A1 (0.71) CYP1A2MEN1KMT2APOLBGAA
SCHEMBL24328063 0.69 NPC1 (0.52) CYP1A2CYP3A4MEN1KMT2APOLB
SCHEMBL27477545 0.67 CYP1A2 (0.43) CYP1A2CYP3A4MEN1KMT2APOLB
SCHEMBL5523767 0.65 CYP1A2 (0.58) CYP1A2CYP3A4MEN1KMT2AGAA
SCHEMBL24327926 0.64 CYP1A2 (0.40) CYP1A2CYP3A4MEN1KMT2AGAA
SCHEMBL24327446 0.64 MTOR (0.48) CA1CA2CA9LMNAMAPT
SCHEMBL29140936 0.64 MTOR (0.78) MEN1KMT2ACA1CA2CA9
SCHEMBL11682405 0.64 HSP90AA1 (0.43) POLBSMN1; SMN2NPC1RAB9AHDAC6
SCHEMBL12585097 0.64 MEN1 (0.79) MEN1KMT2APOLBGAACA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022081984-A1 METHODS AND COMPOUNDS TO TREAT SARS INFECTIONS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-04-21 WO disclosed