SCHEMBL24333397

SCHEMBL24333397

CCc1cccc(OCc2ccccc2)c1S(=O)(=O)NC(=O)c1cc2c(F)cc(N3CCC3)cc2o1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 2/20 0.38
PTGER1 P34995 4/20 0.37
MRGPRX4 Q96LA9 2/20 0.35
PSMD14 O00487 1/20 0.35
USP2 O75604 1/20 0.35
LRRK2 Q5S007 2/20 0.34
ABCB1 P08183 2/20 0.34
ABCG2 Q9UNQ0 2/20 0.34
TP53 P04637 1/20 0.34
NPC1 O15118 1/20 0.34
KDM1A O60341 2/20 0.33
HPGD P15428 1/20 0.33
HTT P42858 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MAOB P27338 1/20 0.33
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29469638 1.00 MMP2 (0.38) MMP2PTGER1MRGPRX4PSMD14USP2
SCHEMBL24333633 0.93 PTGER1 (0.39) MMP2PTGER1MRGPRX4LRRK2ABCB1
SCHEMBL29469636 0.93 PTGER1 (0.39) MMP2PTGER1MRGPRX4LRRK2ABCB1
SCHEMBL24333765 0.90 USP2 (0.36) USP2NPC1HPGDHTTDRD2
SCHEMBL29469721 0.89 SCN9A (0.36)
SCHEMBL24333693 0.89 SCN9A (0.36)
SCHEMBL29469621 0.88 PTGDR (0.36) MMP2TP53NPC1HTT
SCHEMBL24333945 0.87 PTGER1 (0.36) MMP2PTGER1LRRK2KDM1AMAOB
SCHEMBL29469650 0.87 PTGER1 (0.36) MMP2PTGER1LRRK2KDM1AMAOB
SCHEMBL24333958 0.86 ALDH1A1 (0.33) MMP2PSMD14USP2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022081807-A1 SUBSTITUTED ACYL SULFONAMIDES FOR TREATING CANCER THE BROAD INSTITUTE, INC. (US) 2022-04-21 WO disclosed