SCHEMBL2433801

SCHEMBL2433801

CNC(=O)c1c(-c2ccc(F)cc2)nn2ccc(-c3cc(C(=O)N(c4ccccn4)C4CC4)c(OC(F)F)nc3C)c(F)c12

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
CNR2 P34972 2/20 0.32
CNR1 P21554 1/20 0.32
CSNK1D P48730 1/20 0.31
CSNK1E P49674 1/20 0.31
JAK2 O60674 2/20 0.30
JAK1 P23458 2/20 0.30
ABHD6 Q9BV23 1/20 0.30
TRPM8 Q7Z2W7 1/20 0.30
TNF P01375 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1936514 0.83 ALDH1A1 (0.45) ALDH1A1TRPM8
SCHEMBL2469800 0.82 CSNK1D (0.37) ALDH1A1CNR2CNR1CSNK1DCSNK1E
SCHEMBL2464901 0.82 CYP2C8 (0.43) CNR2CNR1
SCHEMBL2468592 0.81 GRM4 (0.36) CNR2CNR1
SCHEMBL2465370 0.79 CYP2C8 (0.40) CNR2CNR1CSNK1DCSNK1E
SCHEMBL2432013 0.75 CSF1R (0.31) CNR2ABHD6
SCHEMBL2470386 0.74 CYP2C8 (0.44) CNR2CNR1CSNK1DCSNK1EABHD6
SCHEMBL2467631 0.74 NPC1 (0.38) CNR2CNR1CSNK1DCSNK1EABHD6
SCHEMBL2468380 0.74 CSNK1D (0.37) CNR2CNR1CSNK1DCSNK1EABHD6
SCHEMBL2467958 0.72 CNR1 (0.38) CNR2CNR1CSNK1DCSNK1EABHD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2545050-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C Bristol-Myers Squibb Company (US) 2013-01-16 EP disclosed
WO-2011112186-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2011-09-15 WO disclosed