SCHEMBL2468592

SCHEMBL2468592

CNC(=O)c1c(-c2ccc(F)cc2)nn2ccc(-c3cc(C(=O)N(c4ncccn4)C4CC4)c(OCC4CCOCC4)nc3C)c(F)c12

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 16/20 0.36
CNR1 P21554 2/20 0.34
CNR2 P34972 1/20 0.34
RIPK1 Q13546 1/20 0.33
GABRA5 P31644 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2467958 0.88 CNR1 (0.38) GRM4CNR1CNR2RIPK1GABRA5
SCHEMBL2468589 0.86 CYP2C8 (0.42) GRM4CNR1CNR2RIPK1
SCHEMBL2464498 0.84 CYP2C8 (0.41) GRM4CNR1CNR2RIPK1
SCHEMBL2433801 0.81 ALDH1A1 (0.36) CNR1CNR2
SCHEMBL2432013 0.77 CSF1R (0.31) CNR2
SCHEMBL2467631 0.73 NPC1 (0.38) CNR1CNR2RIPK1
SCHEMBL2468380 0.73 CSNK1D (0.37) CNR1CNR2RIPK1
SCHEMBL1936514 0.72 ALDH1A1 (0.45)
SCHEMBL2469800 0.71 CSNK1D (0.37) CNR1CNR2RIPK1
SCHEMBL1936635 0.71 TYK2 (0.33) CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2545050-B1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL MYERS SQUIBB CO (US) 2014-08-13 EP claimed
EP-2545050-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C Bristol-Myers Squibb Company (US) 2013-01-16 EP claimed
WO-2011112186-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2011-09-15 WO claimed
EP-2545050-B1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL MYERS SQUIBB CO (US) 2014-08-13 EP disclosed
EP-2545050-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C Bristol-Myers Squibb Company (US) 2013-01-16 EP disclosed
WO-2011112186-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2011-09-15 WO disclosed