SCHEMBL24338701

SCHEMBL24338701

CCOC(=O)c1c(C2CC2)nn2cccc(CO)c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 2/20 0.39
DGAT1 O75907 2/20 0.39
SOAT1 P35610 1/20 0.39
TSHR P16473 3/20 0.39
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.38
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37
DRD2 P14416 1/20 0.37
DRD4 P21917 1/20 0.37
DRD3 P35462 1/20 0.37
ELANE P08246 2/20 0.36
DHODH Q02127 1/20 0.36
HSD17B10 Q99714 2/20 0.36
GAA P10253 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24338716 0.83 MTNR1A (0.38) PDE4DDRD2DRD4
SCHEMBL543886 0.83 PDE4D (0.50) PDE4DALDH1A1LMNACA12CA1
SCHEMBL3226491 0.81 PDE4D (0.42) PDE4DTSHRALDH1A1LMNACA12
SCHEMBL3217956 0.78 KDM4E (0.41) PDE4DTSHRALDH1A1LMNACA12
SCHEMBL6716443 0.75 PDE4D (0.52) PDE4DALDH1A1LMNACA12CA1
SCHEMBL30174407 0.74 MAPK8 (0.37) PDE4DDGAT1SOAT1TSHRALDH1A1
SCHEMBL14684369 0.71 PDE4D (0.43) PDE4DALDH1A1LMNAHSD17B10GAA
SCHEMBL1290595 0.71 DRD2 (0.60) TSHRALDH1A1LMNADRD2DRD4
SCHEMBL29241266 0.70 POLB (0.45) PDE4DLMNAGAATP53MAPT
SCHEMBL3459020 0.69 ALDH1A1 (0.39) ALDH1A1LMNACA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115515956-A Benzimidazole derivative and preparation method and medical application thereof 深圳信立泰药业股份有限公司 2022-12-23 CN disclosed
WO-2022068772-A1 BENZIMIDAZOLE DERIVATIVE, AND PREPARATION METHOD THEREFOR, AND MEDICAL USE THEREOF 深圳信立泰药业股份有限公司 2022-04-07 WO disclosed
WO-2022068772-A1 BENZIMIDAZOLE DERIVATIVE, AND PREPARATION METHOD THEREFOR, AND MEDICAL USE THEREOF 深圳信立泰药业股份有限公司 2022-04-07 WO disclosed