SCHEMBL2434582

SCHEMBL2434582

Cc1cc[c]c(-c2ccc(F)c(F)c2)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 1/20 0.35
NOTUM Q6P988 1/20 0.33
RAPGEF4 Q8WZA2 1/20 0.33
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32
CYP17A1 P05093 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31
PTGS2 P35354 3/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
GAA P10253 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
MAOB P27338 1/20 0.30
HSD17B1 P14061 1/20 0.30
HSD17B2 P37059 1/20 0.30
PTGS1 P23219 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1491043 0.81 ACHE (0.41) NFE2L2ALDH1A1MAOB
SCHEMBL9521923 0.81 NOTUM (0.35) NFE2L2NOTUMCYP17A1CYP11B1CYP11B2
SCHEMBL2431368 0.79 NOTUM (0.34) NOTUMCYP17A1CYP11B1CYP11B2CES2
SCHEMBL102139 0.78 TDP1 (0.36) ALDH1A1CYP1A2MAOB
SCHEMBL3977645 0.77 NOTUM (0.35) NOTUMPTGS2ALDH1A1
SCHEMBL2013006 0.77 ACHE (0.35)
SCHEMBL2154312 0.77 AHR (0.34) NOTUMPTGS2ALDH1A1CYP1A2
SCHEMBL2014176 0.76 ACHE (0.50) NFE2L2NOTUMRAPGEF4ALDH1A1GAA
SCHEMBL2015248 0.75 TRPA1 (0.43) NOTUMCYP11B1CYP11B2PTGS2HSD17B1
SCHEMBL7049757 0.75 ACHE (0.38) ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013182433-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-12-12 WO disclosed
EP-2547687-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-01-23 EP disclosed
EP-2513067-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2012-10-24 EP disclosed
WO-2011113820-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2011-09-22 WO disclosed