SCHEMBL2015248

SCHEMBL2015248

Fc1ccc(-c2[c]ccc(C(F)(F)F)c2)cc1F

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 3/20 0.43
PDE2A O00408 3/20 0.33
KIF11 P52732 5/20 0.33
MPL P40238 1/20 0.33
IDO1 P14902 1/20 0.33
ALOX5AP P20292 2/20 0.32
FEN1 P39748 2/20 0.32
HSD17B1 P14061 1/20 0.32
HSD17B2 P37059 1/20 0.32
NOTUM Q6P988 1/20 0.32
PTGS2 P35354 2/20 0.32
PTGS1 P23219 1/20 0.32
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1690372 0.82 SMN1; SMN2 (0.34) PDE2AKIF11
SCHEMBL8078153 0.82 KIF11 (0.43) KIF11NOTUM
SCHEMBL6246969 0.81 TRPV1 (0.36) KIF11CYP11B1CYP11B2
SCHEMBL10340202 0.81 PTGDR2 (0.38) NOTUMPTGS2PTGS1
SCHEMBL2431368 0.80 NOTUM (0.34) TRPA1HSD17B1HSD17B2NOTUMCYP11B1
SCHEMBL2013705 0.79 RXRA (0.33) PDE2A
SCHEMBL2204411 0.79 NOTUM (0.43) KIF11IDO1NOTUM
SCHEMBL9521923 0.78 NOTUM (0.35) HSD17B1HSD17B2NOTUMPTGS2PTGS1
SCHEMBL2431003 0.78 PTPN1 (0.39) TRPA1HSD17B1HSD17B2CYP11B2
SCHEMBL16055751 0.77 NPBWR1 (0.41) KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784388-B3 BIPHENYLOXYACETIC ACID DERIVATIVES FOR THE TREATMENT OF RESPIRATORY DISEASE ASTRAZENECA AB (SE) 2012-09-05 EP claimed
WO-2013182433-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-12-12 WO disclosed
EP-2547687-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-01-23 EP disclosed
EP-2513067-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2012-10-24 EP disclosed
WO-2011113820-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2011-09-22 WO disclosed
WO-2011073145-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2011-06-23 WO disclosed