SCHEMBL24359063

SCHEMBL24359063

COC[C@@H]1CCCN1CC(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
HDAC1 Q13547 1/20 0.41
ARG1 P05089 2/20 0.40
ARG2 P78540 2/20 0.40
CRHR1 P34998 1/20 0.38
DRD2 P14416 2/20 0.37
HTR2A P28223 2/20 0.37
HTR2C P28335 2/20 0.37
VEGFA P15692 1/20 0.36
EGLN1 Q9GZT9 1/20 0.36
PNP P00491 1/20 0.35
CASP3 P42574 3/20 0.34
CASP7 P55210 3/20 0.34
HTR1D P28221 1/20 0.34
HTR1B P28222 1/20 0.34
ADORA2A P29274 1/20 0.34
TLR7 Q9NYK1 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
DPP4 P27487 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25540249 1.00 HDAC8 (0.41) HDAC8HDAC6HDAC1ARG1ARG2
SCHEMBL24359060 0.89 HDAC8 (0.31) HDAC8HDAC6HDAC1ARG1ARG2
SCHEMBL9283501 0.84 HDAC8 (0.42) HDAC8HDAC6HDAC1ARG1ARG2
SCHEMBL9284738 0.84 HDAC8 (0.42) HDAC8HDAC6HDAC1ARG1ARG2
SCHEMBL12788428 0.84 HDAC8 (0.42) HDAC8HDAC6HDAC1ARG1ARG2
SCHEMBL24731188 0.81 CRHR1 (0.30) CRHR1
SCHEMBL28858890 0.81 ALDH1A1 (0.34) HDAC8HDAC6HDAC1DRD2CASP3
SCHEMBL24359069 0.81 CRHR1 (0.30) CRHR1
SCHEMBL14922679 0.79 ATM (0.40) HRH3
SCHEMBL28283697 0.79 ATM (0.40) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022087624-A1 COMPOUNDS AS RAS INHIBITORS AND USES THEREOF BIOARDIS LLC (US) 2022-04-28 WO disclosed