SCHEMBL243630

SCHEMBL243630

COc1ccc(C2c3ccc(O)cc3OCC2c2ccc(Br)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.54
ESR2 Q92731 5/20 0.54
EDNRB P24530 1/20 0.46
EDNRA P25101 1/20 0.46
ALDH1A1 P00352 1/20 0.42
ALOX15 P16050 2/20 0.42
ALOX12 P18054 2/20 0.42
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
LMNA P02545 1/20 0.39
MAOB P27338 2/20 0.39
CYP3A4 P08684 1/20 0.39
MAOA P21397 1/20 0.39
MGAM O43451 1/20 0.38
POLB P06746 1/20 0.37
RECQL P46063 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30362777 1.00 ESR1 (0.54) ESR1ESR2EDNRBEDNRAALDH1A1
SCHEMBL25892433 1.00 ESR1 (0.54) ESR1ESR2EDNRBEDNRAALDH1A1
SCHEMBL24103125 1.00 ESR1 (0.54) ESR1ESR2EDNRBEDNRAALDH1A1
SCHEMBL15013033 0.93 ESR1 (0.58) ESR1ESR2EDNRBEDNRAALDH1A1
SCHEMBL20831831 0.93 ESR1 (0.58) ESR1ESR2EDNRBEDNRAALDH1A1
SCHEMBL2604720 0.93 ESR1 (0.58) ESR1ESR2EDNRBEDNRAALDH1A1
SCHEMBL239999 0.93 ESR1 (0.58) ESR1ESR2EDNRBEDNRAALDH1A1
SCHEMBL20831829 0.93 ESR1 (0.58) ESR1ESR2EDNRBEDNRAALDH1A1
SCHEMBL15312307 0.93 ESR1 (0.58) ESR1ESR2EDNRBEDNRAALDH1A1
SCHEMBL30362855 0.93 ESR1 (0.58) ESR1ESR2EDNRBEDNRAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 68 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120172424-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY MARSHALL EDWARDS, INC. (US) 2012-07-05 US claimed
US-8080675-B2 Chroman derivatives, medicaments and use in therapy MARSHALL EDWARDS, INC. (US) 2011-12-20 US claimed
EP-1809618-A4 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RES PTY LTD (AU) 2008-11-19 EP claimed
EP-1809618-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY Novogen Research Pty Ltd (AU) 2007-07-25 EP claimed
US-20060074126-A1 Chroman derivatives, medicaments and use in therapy NOVOGEN RESEARCH PTY LTD 2006-04-06 US claimed
WO-2006032086-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RESEARCH PTY LTD (AU) 2006-03-30 WO claimed
US-12414934-B2 Combination therapies Aardvark Therapeutics, Inc. (US) 2025-09-16 US disclosed
WO-2024137472-A2 COMBINATION THERAPIES MEI PHARMA, INC. (US) 2024-06-27 WO disclosed
US-20230233519-A1 COMBINATION THERAPIES Aardvark Therapeutics, Inc. 2023-07-27 US disclosed
US-20230233519-A1 COMBINATION THERAPIES Aardvark Therapeutics, Inc. 2023-07-27 US disclosed
US-20230233519-A1 COMBINATION THERAPIES Aardvark Therapeutics, Inc. 2023-07-27 US disclosed
CN-116139125-A Combination therapy 梅制药公司 2023-05-23 CN disclosed
EP-4164632-A1 COMBINATION THERAPIES MEI Pharma, Inc. (US) 2023-04-19 EP disclosed
WO-2010022467-A1 IMMUNOMODULATING ACTIVITIES NOVOGEN RESEARCH PTY LTD (AU) 2010-03-04 WO disclosed
EP-2120925-A1 METHOD FOR INDUCING AUTOPHAGY Novogen Research Pty. Ltd. (AU) 2009-11-25 EP disclosed
EP-1809618-A4 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RES PTY LTD (AU) 2008-11-19 EP disclosed
WO-2008113100-A1 METHOD FOR INDUCING AUTOPHAGY NOVOGEN RESEARCH PTY LTD (AU) 2008-09-25 WO disclosed
EP-1809618-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY Novogen Research Pty Ltd (AU) 2007-07-25 EP disclosed
US-20060074126-A1 Chroman derivatives, medicaments and use in therapy NOVOGEN RESEARCH PTY LTD 2006-04-06 US disclosed
WO-2006032086-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY NOVOGEN RESEARCH PTY LTD (AU) 2006-03-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12414934-B2 Combination therapies PCK2, PDK1, PCK1 ESR1 2467/4885ESR2 1403/4885EDNRB 2845/4885
US-20230233519-A1 COMBINATION THERAPIES BCL2, BAK1, BCL2L2 ESR1 3784/4885ESR2 2187/4885EDNRB 3424/4885
US-20120172424-A1 CHROMAN DERIVATIVES, MEDICAMENTS AND USE IN THERAPY CDYL, XPA, TP53 ESR1 1699/4885ESR2 1586/4885EDNRB 4204/4885
US-20060074126-A1 Chroman derivatives, medicaments and use in therapy CDYL, XPA, TP53 ESR1 1699/4885ESR2 1586/4885EDNRB 4204/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.