SCHEMBL24364984

SCHEMBL24364984

c1ccc2c(C3CCCCN3)csc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.43
DRD2 P14416 1/20 0.43
CYP2A6 P11509 3/20 0.41
MEN1 O00255 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C19 P33261 2/20 0.41
KMT2A Q03164 2/20 0.41
CHRNA7 P36544 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
POLB P06746 2/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CRHBP P24387 1/20 0.38
CRHR2 Q13324 1/20 0.38
OPRM1 P35372 2/20 0.38
OPRK1 P41145 2/20 0.38
MTNR1A P48039 1/20 0.37
CHRM5 P08912 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28502662 0.95 SLC6A4 (0.43) SLC6A4DRD2CYP2A6MEN1KMT2A
SCHEMBL7993430 0.79 SLC6A4 (0.40) SLC6A4DRD2CYP2A6CYP2D6CHRNA7
SCHEMBL18908547 0.78 SLC6A4 (0.59) SLC6A4DRD2CYP2A6CHRNA7SMN1; SMN2
SCHEMBL30469977 0.77 SLC6A4 (0.43) SLC6A4DRD2CYP2A6CHRNA7SMN1; SMN2
SCHEMBL29081842 0.77 SLC6A4 (0.43) SLC6A4DRD2CYP2A6CHRNA7SMN1; SMN2
SCHEMBL29324945 0.77 SLC6A4 (0.43) SLC6A4DRD2CYP2A6CHRNA7SMN1; SMN2
SCHEMBL24364676 0.77 SLC6A4 (0.43) SLC6A4DRD2CYP2A6CHRNA7SMN1; SMN2
SCHEMBL28509100 0.74 SLC6A2 (0.42) SLC6A4DRD2CYP2A6MEN1CYP2D6
SCHEMBL22252026 0.74 SLC6A4 (0.59) SLC6A4DRD2CYP2A6CHRNA7SMN1; SMN2
SCHEMBL9634176 0.73 KDM1A (0.43) SLC6A4CYP2A6MEN1CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260078117-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS INC (US) 2026-03-19 US disclosed
US-20240228478-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS, INC. 2024-07-11 US disclosed
US-20240228478-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS, INC. 2024-07-11 US disclosed
CN-116568677-A piperidin-1-yl-N-pyridin-3-yl-2-oxoacetamide derivatives useful for the treatment of MTAP deficiency and/or MTA accumulating cancers 探戈医药股份有限公司 2023-08-08 CN disclosed
US-20220127256-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS, INC. 2022-04-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220127256-A1 COMPOUNDS AND METHODS OF USE F12, C1R, ABCG2 SLC6A4 1165/4885DRD2 287/4885CYP2A6 105/4885
US-20240228478-A1 COMPOUNDS AND METHODS OF USE F12, C1R, ABCG2 SLC6A4 1165/4885DRD2 287/4885CYP2A6 105/4885
US-20260078117-A1 COMPOUNDS AND METHODS OF USE NR3C2, ADRA1A, CNR1 SLC6A4 766/4885DRD2 504/4885CYP2A6 30/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.