SCHEMBL24375514

SCHEMBL24375514

COc1ccc(-n2ccc(C)n2)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HTT P42858 1/20 0.44
OGA O60502 1/20 0.42
CHRNB2 P17787 4/20 0.42
CHRNA4 P43681 4/20 0.42
OPRM1 P35372 1/20 0.42
MAPT P10636 2/20 0.40
RAB9A P51151 2/20 0.40
NPC1 O15118 1/20 0.40
ATM Q13315 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CHRNB4 P30926 2/20 0.39
CHRNA3 P32297 2/20 0.39
OXTR P30559 6/20 0.39
AVPR1A P37288 3/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31316711 0.82 CHRNB2 (0.41) MEN1KMT2AOGACHRNB2CHRNA4
SCHEMBL20390801 0.82 CHRNB2 (0.41) MEN1KMT2AOGACHRNB2CHRNA4
SCHEMBL26401548 0.80 HTT (0.50) HTTCHRNB2CHRNA4OPRM1MAPT
SCHEMBL15925373 0.80 CHRNB2 (0.40) MEN1KMT2AOGACHRNB2CHRNA4
SCHEMBL24375517 0.80 FYN (0.48) MEN1KMT2AHTTOGACHRNB2
SCHEMBL15935407 0.79 HTT (0.42) KMT2AHTTMAPTRAB9ANPC1
SCHEMBL20594704 0.77 IRAK4 (0.44) MEN1KMT2AHTTOGACHRNB2
SCHEMBL21840502 0.76 IRAK4 (0.46) MEN1KMT2AHTTCHRNB2CHRNA4
SCHEMBL15832231 0.75 RAB9A (0.41) HTTMAPTRAB9ANPC1ATM
SCHEMBL15935032 0.75 ELOVL1 (0.44) HTTOPRM1MAPTRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3642199-B1 BENZOFURANS AS IRAK4 MODULATORS HOFFMANN LA ROCHE (CH) 2022-04-27 EP disclosed