SCHEMBL24377322

SCHEMBL24377322

CCc1cccn2c(N)nnc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATP4A P20648 1/20 0.37
ATP4B P51164 1/20 0.37
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
TLR8 Q9NR97 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD11B1 P28845 3/20 0.33
NR1I2 O75469 2/20 0.33
GABRA1 P14867 2/20 0.32
GABRB2 P47870 2/20 0.32
KMT2A Q03164 1/20 0.32
LMNA P02545 1/20 0.32
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GLA P06280 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24377487 0.76 ALDH1A1 (0.47) SMN1; SMN2HSD11B1NR1I2KDM4ENPC1
SCHEMBL17437975 0.75 SMN1; SMN2 (0.38) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL24377254 0.71 HSD11B1 (0.48) CYP1A2CYP3A4HSD11B1NR1I2GABRA1
SCHEMBL16158057 0.71 NR3C2 (0.44) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL16158058 0.69 KMT2A (0.37) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL23108726 0.68 CYP1A2 (0.38) ATP4AATP4BCYP1A2CYP3A4CYP2D6
SCHEMBL16157995 0.67 CHEK1 (0.43) MAPK14
SCHEMBL26476504 0.67 ADORA3 (0.47) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL6468439 0.66 TP53 (0.40) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL18231784 0.65 CYP1A2 (0.41) ATP4AATP4BCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022086920-A1 GLUTAMINYL-PEPTIDE CYCLOTRANSFERASE LIKE (QPCTL) PROTEIN INHIBITORS AND USES THEREOF BLACKSMITH MEDICINES, INC. (US) 2022-04-28 WO disclosed