SCHEMBL24378573

SCHEMBL24378573

CC(C)(O)NCCNC(=O)c1cc2nc(Cl)cc(N3CCOCC3)n2n1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
GAA P10253 2/20 0.42
KDM4E B2RXH2 1/20 0.42
GLA P06280 1/20 0.42
CFTR P13569 2/20 0.37
MKNK1 Q9BUB5 3/20 0.36
RAF1 P04049 3/20 0.36
BRAF P15056 3/20 0.36
PARP1 P09874 2/20 0.36
HDAC6 Q9UBN7 1/20 0.35
HPGD P15428 2/20 0.35
TP53 P04637 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
NAPEPLD Q6IQ20 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24378424 0.88 ALDH1A1 (0.42) ALDH1A1GAAKDM4EGLACFTR
SCHEMBL24378656 0.87 ALDH1A1 (0.42) ALDH1A1GAAKDM4EGLACFTR
SCHEMBL22718383 0.78 CNR2 (0.39) ALDH1A1GAAKDM4EGLACFTR
SCHEMBL24378574 0.77 KDM4E (0.40) ALDH1A1GAAKDM4EGLAHPGD
SCHEMBL22718319 0.77 KMO (0.44) ALDH1A1KDM4EHPGDSMN1; SMN2CYP1A2
SCHEMBL27009142 0.75 HPGD (0.43) ALDH1A1GAAKDM4EHPGDTP53
SCHEMBL27009137 0.74 HPGD (0.53) ALDH1A1KDM4EHPGDTP53SMN1; SMN2
SCHEMBL22727800 0.74 CNR2 (0.39) ALDH1A1GAAKDM4EGLACFTR
SCHEMBL13815641 0.74 PIK3CA (0.45) ALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL29547619 0.74 HPGD (0.48) ALDH1A1GAAKDM4EHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022086993-A1 NOVEL INHIBITORS OF PIKFYVE AND METHODS USING SAME TME THERAPEUTICS LLC (US) 2022-04-28 WO disclosed