SCHEMBL243932

SCHEMBL243932

O=C(CBr)Nc1ccc(Cl)cc1

nearest known ligand 0.66

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.59
MEN1 O00255 5/20 0.59
SMN1; SMN2 Q16637 2/20 0.59
LMNA P02545 1/20 0.59
HTT P42858 1/20 0.59
ALDH1A1 P00352 6/20 0.58
POLB P06746 1/20 0.58
NPC1 O15118 2/20 0.56
TSHR P16473 2/20 0.56
RAB9A P51151 1/20 0.56
GAA P10253 1/20 0.56
MAPT P10636 1/20 0.56
HPGD P15428 1/20 0.56
ALOX15 P16050 1/20 0.56
HSD17B10 Q99714 1/20 0.56
P2RX7 Q99572 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.50
GSK3B P49841 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15267699 0.89 KMT2A (0.60) KMT2AMEN1LMNAHTTALDH1A1
SCHEMBL6407780 0.86 KMT2A (0.56) KMT2AMEN1SMN1; SMN2LMNAHTT
SCHEMBL1534196 0.84 TP53 (0.64) KMT2AMEN1SMN1; SMN2LMNAHTT
SCHEMBL28422775 0.81 KMT2A (0.53) KMT2AMEN1SMN1; SMN2LMNAHTT
SCHEMBL2098193 0.81 ALDH1A1 (0.59) KMT2AMEN1SMN1; SMN2LMNAHTT
SCHEMBL2098194 0.81 ALDH1A1 (0.59) KMT2AMEN1SMN1; SMN2LMNAHTT
SCHEMBL16922181 0.81 NPC1 (0.66) KMT2AMEN1SMN1; SMN2LMNAHTT
SCHEMBL1039601 0.81 KMT2A (0.76) KMT2AMEN1SMN1; SMN2LMNAHTT
SCHEMBL7888049 0.81 CYP1A1 (0.60) KMT2AMEN1LMNAALDH1A1POLB
SCHEMBL1503954 0.81 NPC1 (0.66) KMT2AMEN1SMN1; SMN2LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 80 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4102924-A REACTING ACYLAMINO-ARYLS WITH HALO-ARYLS BAYER AKTIENGESELLSCHAFT (DE) 1978-07-25 US claimed
JP-6299097-A None JP disclosed
US-20250270217-A1 IMIDAZ0[1,2-A]PYRIMIDINE-5(1 H)-ONES HAVING A COVALENT WARHEAD AT THE 3-POSITION AS WRN INHIBITORS INCYTE CORPORATION (US) 2025-08-28 US disclosed
US-12371429-B2 Antibiotic resistance-modifying tricyclic heteroaryl compounds and uses thereof RECREO PHARMACEUTICALS LLC (US) 2025-07-29 US disclosed
CN-118459362-A N-aryl-2- (2-hydroxybenzyloxy) acetamides, preparation method and application thereof 湖南科技大学 2024-08-09 CN disclosed
US-20240034727-A1 IMIDAZOLE COMPOUNDS AS INHIBITORS OF ENPP1 Stingray Therapeutics, Inc. 2024-02-01 US disclosed
CN-117003744-A Five-membered and six-membered compound, intermediate, preparation method, composition and application 厦门市博瑞来医药科技有限公司 2023-11-07 CN disclosed
CN-116963733-A Imidazole compounds as ENPP1 inhibitors 斯汀格瑞治疗股份有限公司 2023-10-27 CN disclosed
EP-4255425-A1 IMIDAZOLE COMPOUNDS AS INHIBITORS OF ENPP1 Stingray Therapeutics, Inc. (US) 2023-10-11 EP disclosed
CN-114409657-B 4-aryl (methyl) imidazoline quinoxalinone compound and preparation method and application thereof 湖南科技大学 2023-02-24 CN disclosed
EP-1426364-A1 Imidazole-derivatives as factor Xa inhibitors Aventis Pharma Deutschland GmbH (DE) 2004-06-09 EP disclosed
US-20030199689-A1 New indole derivatives as factor Xa inhibitors SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2003-10-23 US disclosed
WO-2003044014-A1 INDOLE-2-CARBOXAMIDES AS FACTOR XA INHIBITORS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2003-05-30 WO disclosed
EP-1077701-A4 ANTI-VIRAL COMPOUNDS LILLY CO ELI (US) 2002-03-20 EP disclosed
EP-1077701-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 2001-02-28 EP disclosed
JP-2000198771-A PHENYLPYRROLIDINONE DERIVATIVE EISAI CO LTD 2000-07-18 JP disclosed
WO-1999059587-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 1999-11-25 WO disclosed
JP-H06299097-A ANTIFOULING COATING COMPOSITION ISHIHARA SANGYO KAISHA LTD 1994-10-25 JP disclosed
EP-0140271-A2 Iodoacetamides BAYER AG (DE) 1985-05-08 EP disclosed
US-4102924-A REACTING ACYLAMINO-ARYLS WITH HALO-ARYLS BAYER AKTIENGESELLSCHAFT (DE) 1978-07-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12371429-B2 Antibiotic resistance-modifying tricyclic heteroaryl compounds and uses thereof CBR3, CBR1, CYP2B6 KMT2A 1544/4885MEN1 1968/4885SMN1; SMN2 4241/4885
US-20240034727-A1 IMIDAZOLE COMPOUNDS AS INHIBITORS OF ENPP1 ENPP1, PPP1R1B, PPM1B KMT2A 2718/4885MEN1 231/4885SMN1; SMN2 865/4885
US-20250270217-A1 IMIDAZ0[1,2-A]PYRIMIDINE-5(1 H)-ONES HAVING A COVALENT WARHEAD AT THE 3-POSITION AS WRN INHIBITORS WRN, RECQL, BLM KMT2A 1697/4885MEN1 1859/4885SMN1; SMN2 2576/4885
US-20030199689-A1 New indole derivatives as factor Xa inhibitors F5, F12, F2 KMT2A 1093/4885MEN1 1167/4885SMN1; SMN2 4319/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.