SCHEMBL24439731

SCHEMBL24439731

Cc1nc(-c2sc(F)cc2CO)ccc1OC1CCCCC1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.33
RECQL P46063 1/20 0.32
PDE4D Q08499 3/20 0.32
KMO O15229 1/20 0.32
PDE4A P27815 4/20 0.32
PDE4B Q07343 3/20 0.32
PDE4C Q08493 2/20 0.32
FPR2 P25090 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
NPY1R P25929 1/20 0.31
NPY2R P49146 1/20 0.31
EPHX2 P34913 1/20 0.31
LPAR1 Q92633 1/20 0.31
FFAR4 Q5NUL3 1/20 0.31
PPARD Q03181 1/20 0.31
S1PR5 Q9H228 1/20 0.31
CSNK2A1 P68400 1/20 0.30
APP P05067 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24441059 0.89 CSNK2A1 (0.38) RIPK1PDE4DKMOPDE4AMEN1
SCHEMBL29672295 0.87 KMO (0.36) RECQLPDE4DKMOPDE4APDE4B
SCHEMBL24439734 0.87 KMO (0.36) RECQLPDE4DKMOPDE4APDE4B
SCHEMBL28744725 0.85 LPAR1 (0.47) PDE4DPDE4APDE4BPDE4CLPAR1
SCHEMBL29672126 0.84 LPAR1 (0.33) RIPK1RECQLPDE4DKMOPDE4A
SCHEMBL24439314 0.84 LPAR1 (0.33) RIPK1RECQLPDE4DKMOPDE4A
SCHEMBL29517377 0.84 LPAR1 (0.41) RIPK1PDE4DPDE4APDE4BPDE4C
SCHEMBL24439730 0.84 LPAR1 (0.41) RIPK1PDE4DPDE4APDE4BPDE4C
SCHEMBL24439618 0.84 LPAR1 (0.41) RIPK1PDE4DPDE4APDE4BPDE4C
SCHEMBL24439382 0.81 SLCO1B1 (0.40) RIPK1LPAR1FFAR4PPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022100623-A1 NITROGEN-SUBSTITUTED HETEROCYCLIC THIOPHENE COMPOUNDS AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-05-19 WO disclosed
WO-2022100624-A1 OXY-SUBSTITUTED AMINOCARBONATE THIOPHENE-BASED COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-05-19 WO disclosed