SCHEMBL24445679

SCHEMBL24445679

C/C(=N\O)c1ccc(F)cc1F

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.52
CES1 P23141 3/20 0.52
ESR1 P03372 2/20 0.47
ESR2 Q92731 2/20 0.47
MGLL Q99685 1/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
MAPT P10636 5/20 0.42
ALDH1A1 P00352 4/20 0.42
POLB P06746 1/20 0.42
ALOX12 P18054 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
KDM4E B2RXH2 2/20 0.42
MAPK1 P28482 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CA3 P07451 1/20 0.37
CA6 P23280 1/20 0.37
CA5A P35218 1/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18567683 0.82 CES2 (0.50) CES2CES1MEN1KMT2AMAPT
SCHEMBL8181697 0.82 ESR1 (0.50) CES2CES1ESR1ESR2MGLL
SCHEMBL8221493 0.82 ESR1 (0.50) CES2CES1ESR1ESR2MGLL
SCHEMBL13636405 0.82 ESR1 (0.46) CES2CES1ESR1ESR2MGLL
SCHEMBL30690133 0.82 ESR1 (0.50) CES2CES1ESR1ESR2MGLL
SCHEMBL1345659 0.80 MEN1 (0.43) CES2CES1ESR1ESR2MGLL
SCHEMBL1345658 0.80 MEN1 (0.43) CES2CES1ESR1ESR2MGLL
SCHEMBL28905087 0.80 DGAT1 (0.52) ESR1ESR2MGLLMEN1KMT2A
SCHEMBL15761173 0.79 CES2 (0.47) CES2CES1ESR1ESR2MGLL
SCHEMBL6814924 0.79 CES2 (0.47) CES2CES1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3587412-B1 FXR (NR1H4) MODULATING COMPOUNDS GILEAD SCIENCES INC (US) 2022-05-25 EP disclosed