SCHEMBL24446325

SCHEMBL24446325

Cc1ccc2c(c1)SC(C)C2C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.40
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
EPHX2 P34913 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ACHE P22303 1/20 0.33
CYP1A2 P05177 2/20 0.32
CYP2A6 P11509 2/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
ALOX15 P16050 1/20 0.31
ALOX12 P18054 1/20 0.31
BRCA1 P38398 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13894961 0.78 CHRNB2 (0.35) CHRNB2CHRNA4MEN1KMT2AACHE
SCHEMBL14641002 0.78 HTR2C (0.41) HTR2CCHRNB2CHRNA4MEN1KMT2A
SCHEMBL13070499 0.76 ACHE (0.38) HTR2CCHRNB2CHRNA4EPHX2MEN1
SCHEMBL28302528 0.72 KDM4E (0.31)
SCHEMBL10364335 0.71 MEN1 (0.35) HTR2CMEN1KMT2AACHECYP1A2
SCHEMBL24857876 0.71 MEN1 (0.35) HTR2CMEN1KMT2AACHECYP1A2
SCHEMBL12240339 0.69 ACHE (0.42) EPHX2ACHECA1CA2HPGD
SCHEMBL12240335 0.69 ACHE (0.42) EPHX2ACHECA1CA2HPGD
SCHEMBL7920994 0.69 CHRNB2 (0.35) HTR2CCHRNB2CHRNA4EPHX2MEN1
SCHEMBL15582403 0.69 HSD11B1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3097078-B1 PYRIDINES AND PYRIMIDINES AND USE THEREOF PURDUE PHARMA LP (US) 2022-05-25 EP disclosed