Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | ATP1A1 | P05023 | 1/20 | 0.55 |
| ▸ | ATP1B1 | P05026 | 1/20 | 0.55 |
| ▸ | ATP1A3 | P13637 | 1/20 | 0.55 |
| ▸ | ATP1B2 | P14415 | 1/20 | 0.55 |
| ▸ | ATP1A2 | P50993 | 1/20 | 0.55 |
| ▸ | ATP1B3 | P54709 | 1/20 | 0.55 |
| ▸ | FXYD2 | P54710 | 1/20 | 0.55 |
| ▸ | ATP1A4 | Q13733 | 1/20 | 0.55 |
| ▸ | MAPT | P10636 | 3/20 | 0.45 |
| ▸ | MEN1 | O00255 | 1/20 | 0.43 |
| ▸ | KMT2A | Q03164 | 1/20 | 0.43 |
| ▸ | SCN5A | Q14524 | 5/20 | 0.43 |
| ▸ | SCN10A | Q9Y5Y9 | 6/20 | 0.43 |
| ▸ | KCNH2 | Q12809 | 3/20 | 0.43 |
| ▸ | SCN1A | P35498 | 1/20 | 0.43 |
| ▸ | SCN9A | Q15858 | 1/20 | 0.43 |
| ▸ | SCN2A | Q99250 | 1/20 | 0.43 |
| ▸ | SCN8A | Q9UQD0 | 1/20 | 0.43 |
| ▸ | TDP2 | O95551 | 1/20 | 0.42 |
| ▸ | POLB | P06746 | 1/20 | 0.41 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL24460279 | 0.80 | ATP1A1 (0.43) | ATP1A1ATP1B1ATP1A3ATP1B2ATP1A2 | |
| SCHEMBL14077014 | 0.76 | GAA (0.54) | ATP1A1ATP1B1ATP1A3ATP1B2ATP1A2 | |
| SCHEMBL19973142 | 0.74 | ATP1A1 (0.47) | ATP1A1ATP1B1ATP1A3ATP1B2ATP1A2 | |
| SCHEMBL20075887 | 0.74 | GSK3B (0.48) | MAPTMEN1KMT2APOLBTP53 | |
| SCHEMBL19981228 | 0.74 | ATP1A1 (0.45) | ATP1A1ATP1B1ATP1A3ATP1B2ATP1A2 | |
| SCHEMBL22845298 | 0.73 | POLB (0.45) | MAPTPOLBTP53GAAGSK3B | |
| SCHEMBL14077000 | 0.73 | USP2 (0.66) | ATP1A1ATP1B1ATP1A3ATP1B2ATP1A2 | |
| SCHEMBL12492258 | 0.73 | TP53 (0.51) | MAPTMEN1KMT2ATP53GAA | |
| SCHEMBL26361711 | 0.73 | SCN5A (0.56) | ATP1A1ATP1B1ATP1A3ATP1B2ATP1A2 | |
| SCHEMBL12721184 | 0.72 | CYP1A2 (0.63) | ATP1A1ATP1B1ATP1A3ATP1B2ATP1A2 |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| WO-2022108849-A1 | HETEROCYCLIC COMPOUNDS AS THERAPEUTIC AGENTS | ARISAN THERAPEUTICS INC. (US) | 2022-05-27 | — | — | WO | disclosed |