SCHEMBL24460464

SCHEMBL24460464

COc1cc2ncc(C)n2cc1Br

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.39
MTOR P42345 1/20 0.39
RIPK2 O43353 14/20 0.38
MC4R P32245 1/20 0.35
AXL P30530 1/20 0.35
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
ALOX12 P18054 1/20 0.34
NFKB1 P19838 1/20 0.34
RAB9A P51151 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
LYN P07948 3/20 0.33
LCK P06239 2/20 0.33
TGFBR1 P36897 1/20 0.33
SUV39H2 Q9H5I1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24393296 0.84 NRAS (0.39) PIK3CAMTORRIPK2ALDH1A1LYN
SCHEMBL19781567 0.82 PIK3CA (0.38) PIK3CAMTORRIPK2AXLLYN
SCHEMBL19781784 0.79 TRPA1 (0.34) KDM4ENPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL25383907 0.78 RIPK2 (0.38) PIK3CAMTORRIPK2SUV39H2
SCHEMBL25384458 0.78 PRKDC (0.39) PIK3CAMTORRIPK2LYNSUV39H2
SCHEMBL31356618 0.78 RIPK2 (0.38) PIK3CAMTORRIPK2AXLLYN
SCHEMBL20985980 0.77 TGFBR1 (0.34) KDM4ENPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL24975882 0.75 RIPK2 (0.39) RIPK2LYNLCK
SCHEMBL31356594 0.75 RIPK2 (0.36) PIK3CAMTORRIPK2AXLLYN
SCHEMBL25148947 0.74 POLB (0.40) RIPK2KDM4ELYNLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022108849-A1 HETEROCYCLIC COMPOUNDS AS THERAPEUTIC AGENTS ARISAN THERAPEUTICS INC. (US) 2022-05-27 WO disclosed