SCHEMBL24463595

SCHEMBL24463595

Cn1c(C2CC2)nc2cc(I)ccc21

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 10/20 0.41
HTR2B P41595 1/20 0.39
TAAR1 Q96RJ0 1/20 0.38
USP30 Q70CQ3 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
JAK2 O60674 2/20 0.37
JAK1 P23458 2/20 0.37
TYK2 P29597 2/20 0.37
JAK3 P52333 2/20 0.37
APOBEC3A P31941 1/20 0.37
APOBEC3G Q9HC16 1/20 0.37
MCHR1 Q99705 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3574868 0.81 KDM4E (0.47) PDE10AHTR2BTAAR1USP30JAK2
SCHEMBL24463619 0.80 CNR2 (0.46) JAK2JAK1TYK2JAK3
SCHEMBL5851500 0.76 TAAR1 (0.60) PDE10AHTR2BTAAR1TLR7APOBEC3A
SCHEMBL24463602 0.75 ALOX15 (0.40) PDE10ATLR7MCHR1
SCHEMBL3566734 0.75 ALDH1A1 (0.54) APOBEC3AAPOBEC3G
SCHEMBL17561688 0.74 KDM4E (0.55)
SCHEMBL25678221 0.74 ALDH1A1 (0.53) PDE10ATAAR1USP30TLR7JAK2
SCHEMBL25680318 0.74 TLR7 (0.47) PDE10AHTR2BTAAR1USP30TLR7
SCHEMBL10268288 0.73 HTR3E (0.45) PDE10AHTR2BMCHR1
SCHEMBL24463198 0.73 CLK4 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116057045-A Fibroblast growth factor receptor kinase inhibitors 金耐特生物制药公司 2023-05-02 CN disclosed
US-11345681-B1 Inhibitors of fibroblast growth factor receptor kinases KINNATE BIOPHARMA INC. (US) 2022-05-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11345681-B1 Inhibitors of fibroblast growth factor receptor kinases FGFR1, FGFR2, FGFR3 PDE10A 3103/4885HTR2B 4216/4885TAAR1 4256/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.