SCHEMBL24470813

SCHEMBL24470813

CCOC(=O)c1c(C)oc2ccc(OC3CCc4ccccc43)cc12

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.61
ALDH1A1 P00352 6/20 0.54
LMNA P02545 3/20 0.54
MAPK1 P28482 2/20 0.54
KDM4E B2RXH2 6/20 0.53
L3MBTL1 Q9Y468 5/20 0.53
MAPT P10636 3/20 0.53
POLB P06746 2/20 0.53
HIF1A Q16665 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
TSHR P16473 1/20 0.53
HTT P42858 1/20 0.51
HPGD P15428 3/20 0.48
FFAR1 O14842 2/20 0.48
NPSR1 Q6W5P4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29713112 1.00 PTGS2 (0.61) PTGS2ALDH1A1LMNAMAPK1KDM4E
SCHEMBL29713157 0.89 SLC26A4 (0.52) PTGS2LMNAL3MBTL1POLBHTT
SCHEMBL24470883 0.89 SLC26A4 (0.52) PTGS2LMNAL3MBTL1POLBHTT
SCHEMBL12019229 0.78 FFAR1 (0.59) ALDH1A1LMNAMAPK1KDM4EMAPT
SCHEMBL12019248 0.78 FFAR1 (0.51) MAPTPOLBFFAR1
SCHEMBL31604936 0.77 PTGS2 (0.63) PTGS2ALDH1A1LMNAMAPK1KDM4E
SCHEMBL26676604 0.76 ALDH1A1 (0.68) PTGS2ALDH1A1LMNAMAPK1KDM4E
SCHEMBL28654740 0.75 PTGS2 (0.85) PTGS2ALDH1A1LMNAMAPK1KDM4E
SCHEMBL26676599 0.74 ALDH1A1 (0.65) PTGS2ALDH1A1LMNAMAPK1KDM4E
SCHEMBL26676551 0.74 ALDH1A1 (0.65) PTGS2ALDH1A1LMNAMAPK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116761796-A Aryl derivatives for the treatment of TRPM3 mediated disorders 勒芬天主教大学 2023-09-15 CN disclosed
WO-2022112345-A1 ARYL DERIVATIVES FOR TREATING TRPM3 MEDIATED DISORDERS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2022-06-02 WO disclosed