SCHEMBL2447397

SCHEMBL2447397

NC(=O)C1(Cc2ccccc2)CNCCO1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 12/20 0.39
SLC6A4 P31645 12/20 0.39
SLC6A3 Q01959 12/20 0.39
CYP2D6 P10635 6/20 0.39
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
ADAM17 P78536 1/20 0.34
KMT2A Q03164 1/20 0.33
LMNA P02545 1/20 0.33
ALPI P09923 1/20 0.33
PKM P14618 1/20 0.33
PTGS1 P23219 1/20 0.33
XIAP P98170 1/20 0.33
SLC7A5 Q01650 1/20 0.33
CYP3A4 P08684 1/20 0.32
HSD11B1 P28845 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5841607 0.88 SLC6A2 (0.39) SLC6A2SLC6A4SLC6A3CYP2D6KMT2A
SCHEMBL16296491 0.77 PPARG (0.36) MAOAMAOBADAM17KMT2ALMNA
SCHEMBL27788413 0.77 MAOA (0.40) CYP2D6MAOAMAOB
SCHEMBL28012199 0.75 DDB1 (0.41) SLC6A2SLC6A3KMT2ALMNA
SCHEMBL28326929 0.73 KDM4E (0.34) KMT2A
SCHEMBL8862591 0.72 ALPI (0.44) SLC6A2SLC6A4SLC6A3ALPIPKM
SCHEMBL20236439 0.72 HDAC8 (0.37) SLC6A2SLC6A4SLC6A3MAOAKMT2A
SCHEMBL2447412 0.72 HTR2A (0.39) SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL9528556 0.72 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3CYP2D6MAOA
SCHEMBL4557427 0.71 ALDH1A1 (0.35) SLC6A2SLC6A4SLC6A3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2362775-A1 CHEMICAL COMPOUNDS GlaxoSmithKline LLC (US) 2011-09-07 EP disclosed
WO-2010059658-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-05-27 WO disclosed