SCHEMBL2443035

SCHEMBL2443035

CCOc1c(Cl)cc(-c2csc(NC(=O)CBr)n2)cc1Cl

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.49
ABL1 P00519 5/20 0.48
TRPA1 O75762 4/20 0.48
PI4KB Q9UBF8 1/20 0.47
CLK1 P49759 1/20 0.46
PARP1 P09874 1/20 0.46
LMNA P02545 2/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
MAPK1 P28482 1/20 0.44
KMT2A Q03164 1/20 0.44
CYP3A4 P08684 1/20 0.43
ROCK1 Q13464 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15580544 0.93 TRPA1 (0.50) MAPTABL1TRPA1PI4KBRAB9A
SCHEMBL2450859 0.91 TRPA1 (0.48) MAPTABL1TRPA1PI4KBCLK1
SCHEMBL2450980 0.90 RAB9A (0.47) MAPTABL1TRPA1PI4KBCLK1
SCHEMBL13570204 0.89 TRPA1 (0.47) MAPTABL1TRPA1PI4KBCLK1
SCHEMBL480411 0.88 TRPA1 (0.58) MAPTABL1TRPA1PI4KBCLK1
SCHEMBL480792 0.88 TRPA1 (0.61) MAPTABL1TRPA1PI4KBCLK1
SCHEMBL2453455 0.86 TRPA1 (0.49) MAPTABL1TRPA1PI4KBCLK1
SCHEMBL2443409 0.85 ABL1 (0.47) MAPTABL1TRPA1PI4KBCLK1
SCHEMBL2447447 0.85 ABL1 (0.47) MAPTABL1TRPA1PI4KBCLK1
SCHEMBL10139184 0.84 TRPA1 (0.55) MAPTABL1TRPA1PI4KBCLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011114184-A1 AMIDES OF HETEROCYCLIC COMPOUNDS AS TRPA1 INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2011-09-22 WO disclosed
WO-2011114184-A1 AMIDES OF HETEROCYCLIC COMPOUNDS AS TRPA1 INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2011-09-22 WO disclosed