SCHEMBL2448685

SCHEMBL2448685

Cc1cc(N2CCOC[C@H]2C)nc(N)n1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 2/20 0.61
CRHR2 Q13324 2/20 0.61
PDPK1 O15530 2/20 0.54
ROCK1 Q13464 2/20 0.54
AURKB Q96GD4 2/20 0.54
AURKA O14965 1/20 0.54
ATR Q13535 8/20 0.52
ATRIP Q8WXE1 8/20 0.52
CHEK1 O14757 7/20 0.52
PDCD1 Q15116 7/20 0.52
CD274 Q9NZQ7 7/20 0.52
SMN1; SMN2 Q16637 1/20 0.49
HRH3 Q9Y5N1 3/20 0.48
PIK3CA P42336 3/20 0.46
MTOR P42345 3/20 0.46
HRH4 Q9H3N8 1/20 0.44
PIK3CD O00329 2/20 0.44
PIK3R1 P27986 1/20 0.44
PIK3CB P42338 1/20 0.44
PIK3CG P48736 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21516848 0.92 CRHBP (0.55) CRHBPCRHR2PDPK1ROCK1AURKB
SCHEMBL21516206 0.92 CRHBP (0.55) CRHBPCRHR2PDPK1ROCK1AURKB
SCHEMBL3083698 0.91 PDPK1 (0.58) CRHBPCRHR2PDPK1ROCK1AURKB
SCHEMBL1318430 0.84 CYP1A2 (0.60) PDPK1ROCK1AURKBAURKAATR
SCHEMBL20797863 0.82 ATR (0.48) ATRATRIPCHEK1PDCD1CD274
SCHEMBL2513264 0.82 ATR (0.48) ATRATRIPCHEK1PDCD1CD274
SCHEMBL2450233 0.82 CRHBP (0.57) CRHBPCRHR2PDPK1ROCK1AURKB
SCHEMBL22873612 0.80 ATR (0.49) ATRATRIPCHEK1PDCD1CD274
SCHEMBL24175032 0.79 ATR (0.48) ATRATRIPCHEK1PDCD1CD274
SCHEMBL5791956 0.79 CRHBP (0.55) CRHBPCRHR2PDPK1AURKBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2362775-A1 CHEMICAL COMPOUNDS GlaxoSmithKline LLC (US) 2011-09-07 EP disclosed