SCHEMBL2448801

SCHEMBL2448801

NC[C@@H]1[C@H]2CCC[C@H]2CN1C(=O)c1ccccc1-c1ccc(F)cc1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 14/20 0.50
HCRTR2 O43614 10/20 0.46
MLNR O43193 4/20 0.40
CYP3A4 P08684 3/20 0.40
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
CDK4 P11802 1/20 0.39
CCND1 P24385 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2447697 0.92 HCRTR1 (0.57) HCRTR1HCRTR2
SCHEMBL15175749 0.90 HCRTR1 (0.59) HCRTR1HCRTR2
SCHEMBL3415834 0.88 HCRTR1 (0.46) HCRTR1HCRTR2MLNRCYP3A4SLC6A4
SCHEMBL2925288 0.88 HCRTR1 (0.46) HCRTR1HCRTR2MLNRCYP3A4SLC6A4
SCHEMBL2448798 0.85 HCRTR1 (0.46) HCRTR1HCRTR2MLNRCYP3A4SLC6A4
SCHEMBL2448800 0.85 HCRTR1 (0.46) HCRTR1HCRTR2MLNRCYP3A4SLC6A4
SCHEMBL2445627 0.83 HCRTR1 (0.49) HCRTR1HCRTR2CDK4CCND1
SCHEMBL2448756 0.83 HCRTR1 (0.43) HCRTR1HCRTR2MLNRCYP3A4SLC6A4
SCHEMBL2444050 0.81 HCRTR1 (0.47) HCRTR1HCRTR2
SCHEMBL2930541 0.79 HCRTR1 (0.46) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2164847-B1 3-AZA-BICYCLO[3.3.0]OCTANE COMPOUNDS ACTELION PHARMACEUTICALS LTD (CH) 2011-09-14 EP claimed