SCHEMBL24493582

SCHEMBL24493582

CN1CCC(COc2cc(CNN)ccn2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.40
APAF1 O14727 1/20 0.38
CASP3 P42574 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CXCR1 P25024 1/20 0.37
LRRK2 Q5S007 1/20 0.36
EGFR P00533 1/20 0.36
ACACB O00763 3/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
LOX P28300 2/20 0.36
LOXL2 Q9Y4K0 2/20 0.36
SLC6A4 P31645 2/20 0.36
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
CDC42BPB Q9Y5S2 1/20 0.35
PDPK1 O15530 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24493583 0.89 HRH3 (0.40) HRH3APAF1CASP3SENP8SENP7
SCHEMBL30578250 0.86 LOXL2 (0.51) HRH3CXCR1MAOAMAOBLOX
SCHEMBL429671 0.86 LOXL2 (0.51) HRH3CXCR1MAOAMAOBLOX
SCHEMBL427054 0.79 HRH3 (0.44) HRH3CXCR1EGFRMAOAMAOB
SCHEMBL27095942 0.78 APAF1 (0.37) HRH3APAF1CASP3SENP8SENP7
SCHEMBL24493350 0.78 APAF1 (0.41) HRH3APAF1CASP3SENP8SENP7
SCHEMBL24493315 0.78 MRGPRX1 (0.47) ROCK2ROCK1
SCHEMBL30578229 0.78 APAF1 (0.41) HRH3APAF1CASP3SENP8SENP7
SCHEMBL30578216 0.78 MRGPRX1 (0.47) ROCK2ROCK1
SCHEMBL448816 0.78 EGFR (0.40) HRH3CXCR1LRRK2EGFRACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022118016-A2 ENZYME INHIBITORS KALVISTA PHARMACEUTICALS LIMITED (GB) 2022-06-09 WO disclosed