SCHEMBL24497809

SCHEMBL24497809

CCC(CC)OCc1ncc(C)cc1Br

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C19 P33261 1/20 0.30
PRKAG1 P54619 1/20 0.30
PRKAA1 Q13131 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
PRKAB1 Q9Y478 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28207201 0.80 MAPT (0.34) TDP1KDM4EALDH1A1MAPTHPGD
SCHEMBL24497808 0.72 CCR1 (0.35) TDP1KDM4EALDH1A1CYP1A2HDAC6
SCHEMBL31527644 0.71 CCR1 (0.34) TDP1KDM4EALDH1A1MAPTHPGD
Hydrochloric Acid SCHEMBL20767152 0.69 NOS3 (0.38) CYP1A2
SCHEMBL31569231 0.67 CSNK2A1 (0.34) KDM4EALDH1A1MAPT
SCHEMBL1591485 0.66 SLC13A5 (0.40) TDP1KDM4EALDH1A1MAPTHPGD
SCHEMBL30391135 0.66 AGBL2 (0.51) TDP1KDM4EALDH1A1MAPTL3MBTL1
SCHEMBL25168224 0.66 AGBL2 (0.51) TDP1KDM4EALDH1A1MAPTL3MBTL1
SCHEMBL25465424 0.64 ALOX5AP (0.33)
SCHEMBL10703428 0.64 CXCR4 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022119888-A1 3-HETEROARYL PYRROLIDINE AND PIPERIDINE OREXIN RECEPTOR AGONISTS MERCK SHARP & DOHME CORP. (US) 2022-06-09 WO disclosed