SCHEMBL28207201

SCHEMBL28207201

Cc1cnc(COCc2ncc(C)cc2Br)c(Br)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.34
L3MBTL1 Q9Y468 6/20 0.34
TDP1 Q9NUW8 4/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C19 P33261 2/20 0.34
CCR1 P32246 2/20 0.33
CCR5 P51681 2/20 0.33
CCR8 P51685 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
PRKAG1 P54619 1/20 0.33
PRKAA1 Q13131 1/20 0.33
PRKAB1 Q9Y478 1/20 0.33
KDM4E B2RXH2 3/20 0.33
LMNA P02545 2/20 0.33
HPGD P15428 3/20 0.33
ALDH1A1 P00352 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24497809 0.80 TDP1 (0.32) MAPTL3MBTL1TDP1CYP1A2CYP2D6
SCHEMBL24497808 0.79 CCR1 (0.35) TDP1CYP1A2CCR1CCR5CCR8
SCHEMBL31527644 0.78 CCR1 (0.34) MAPTL3MBTL1TDP1CYP1A2CCR1
Hydrochloric Acid SCHEMBL20767152 0.76 NOS3 (0.38) CYP1A2CCR1CCR5CCR8NOS3
SCHEMBL31569231 0.73 CSNK2A1 (0.34) MAPTCCR1CCR5CCR8NOS3
SCHEMBL25168224 0.72 AGBL2 (0.51) MAPTL3MBTL1TDP1KDM4EALDH1A1
SCHEMBL30391135 0.72 AGBL2 (0.51) MAPTL3MBTL1TDP1KDM4EALDH1A1
SCHEMBL10703428 0.71 CXCR4 (0.36) NOS3NOS1NOS2
SCHEMBL762914 0.69
SCHEMBL31180717 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110177551-A HETEROCYCLIC MODULATORS OF LIPID SYNTHESIS 3-V生物科学股份有限公司 2019-08-27 CN disclosed
CN-105001225-B The heterocyclic modulators of lipid synthesis 3-V 生物科学公司 2018-04-06 CN disclosed