SCHEMBL24499463

SCHEMBL24499463

COc1ccc(Br)cc1NC(=O)CBr

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.55
MEN1 O00255 5/20 0.55
NPSR1 Q6W5P4 1/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
MAPT P10636 4/20 0.52
ALDH1A1 P00352 4/20 0.51
TSHR P16473 2/20 0.51
APAF1 O14727 2/20 0.51
POLB P06746 2/20 0.51
GRK2 P25098 2/20 0.51
CTDSP1 Q9GZU7 2/20 0.51
PSMD14 O00487 1/20 0.51
BCL2L1 Q07817 1/20 0.51
MCL1 Q07820 1/20 0.51
KCNT1 Q5JUK3 1/20 0.51
GAA P10253 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
KDM4E B2RXH2 1/20 0.49
S100A4 P26447 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21765898 0.83 SMN1; SMN2 (0.57) KMT2AMEN1NPSR1SMN1; SMN2MAPT
SCHEMBL2374142 0.83 MEN1 (0.80) KMT2AMEN1NPSR1SMN1; SMN2MAPT
SCHEMBL2322923 0.82 KMT2A (0.53) KMT2AMEN1NPSR1SMN1; SMN2MAPT
SCHEMBL14721362 0.82 ALDH1A1 (0.52) KMT2AMEN1NPSR1SMN1; SMN2MAPT
SCHEMBL30362093 0.82 LTB4R (0.64) KMT2AMEN1NPSR1SMN1; SMN2ALDH1A1
Hydrochloric Acid SCHEMBL9487751 0.82 RAD52 (0.62) KMT2AMEN1NPSR1SMN1; SMN2MAPT
SCHEMBL15754270 0.82 LTB4R (0.64) KMT2AMEN1NPSR1SMN1; SMN2ALDH1A1
SCHEMBL3880123 0.81 MAPT (0.51) KMT2AMEN1NPSR1SMN1; SMN2MAPT
SCHEMBL1241796 0.81 KMT2A (0.51) KMT2AMEN1NPSR1SMN1; SMN2MAPT
SCHEMBL24825616 0.79 CYP1A2 (0.53) KMT2AMEN1NPSR1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240034727-A1 IMIDAZOLE COMPOUNDS AS INHIBITORS OF ENPP1 Stingray Therapeutics, Inc. 2024-02-01 US disclosed
CN-116963733-A Imidazole compounds as ENPP1 inhibitors 斯汀格瑞治疗股份有限公司 2023-10-27 CN disclosed
EP-4255425-A1 IMIDAZOLE COMPOUNDS AS INHIBITORS OF ENPP1 Stingray Therapeutics, Inc. (US) 2023-10-11 EP disclosed
WO-2022119928-A1 IMIDAZOLE COMPOUNDS AS INHIBITORS OF ENPP1 Stingray Therapeutics, Inc. (US) 2022-06-09 WO disclosed
WO-2022119928-A1 IMIDAZOLE COMPOUNDS AS INHIBITORS OF ENPP1 Stingray Therapeutics, Inc. (US) 2022-06-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240034727-A1 IMIDAZOLE COMPOUNDS AS INHIBITORS OF ENPP1 ENPP1, PPP1R1B, PPM1B KMT2A 2718/4885MEN1 231/4885NPSR1 4286/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.