SCHEMBL2450367

SCHEMBL2450367

Cc1ccc(CNC(=O)C2CCCNC2)cc1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.56
ALDH1A1 P00352 7/20 0.55
SMN1; SMN2 Q16637 3/20 0.55
USP2 O75604 2/20 0.55
TSHR P16473 2/20 0.55
RAB9A P51151 2/20 0.54
HPGD P15428 2/20 0.51
KDM4E B2RXH2 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.48
POLB P06746 1/20 0.48
CYP3A4 P08684 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17476862 0.87 ALDH1A1 (0.54) HTR2CALDH1A1SMN1; SMN2USP2TSHR
SCHEMBL29542631 0.87 ALDH1A1 (0.57) ALDH1A1TSHRHPGDPOLB
SCHEMBL2444405 0.86 ALDH1A1 (0.70) HTR2CALDH1A1SMN1; SMN2USP2HPGD
SCHEMBL4434645 0.86 ALDH1A1 (0.70) HTR2CALDH1A1SMN1; SMN2USP2HPGD
SCHEMBL2447403 0.86 ALDH1A1 (0.73) HTR2CALDH1A1SMN1; SMN2TSHRRAB9A
SCHEMBL13745623 0.86 HTR2C (0.53) HTR2CALDH1A1SMN1; SMN2USP2RAB9A
Hydrochloric Acid SCHEMBL694838 0.85 HTR2C (0.52) HTR2CALDH1A1SMN1; SMN2USP2TSHR
SCHEMBL10195738 0.84 ALDH1A1 (0.66) ALDH1A1SMN1; SMN2USP2TSHRRAB9A
SCHEMBL29542019 0.84 HTR2C (0.53) HTR2CALDH1A1SMN1; SMN2USP2HPGD
SCHEMBL21541003 0.83 HTR2C (0.62) HTR2CALDH1A1SMN1; SMN2USP2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2600874-A1 PYRIMIDINE COMPOUNDS THAT INHIBIT ANAPLASTIC LYMPHOMA KINASE Amgen, Inc (US) 2013-06-12 EP disclosed
WO-2011143033-A1 PYRIMIDINE COMPOUNDS THAT INHIBIT ANAPLASTIC LYMPHOMA KINASE AMGEN INC. (US) 2011-11-17 WO disclosed
EP-2362775-A1 CHEMICAL COMPOUNDS GlaxoSmithKline LLC (US) 2011-09-07 EP disclosed