SCHEMBL24510481

SCHEMBL24510481

COC(=O)[C@@]12CNCC[C@@H]1C(=O)NC2

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.31
KDM4E B2RXH2 3/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
KMT2A Q03164 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
HTT P42858 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29693908 1.00 POLB (0.31) POLBKDM4EMEN1ALDH1A1CYP1A2
SCHEMBL24510939 0.78
SCHEMBL13537412 0.73 EPHX1 (0.31)
SCHEMBL24510480 0.68 OPRM1 (0.30)
SCHEMBL24510335 0.68 OPRM1 (0.30)
SCHEMBL24510522 0.68 OPRM1 (0.30)
SCHEMBL4748053 0.67 GAA (0.31)
Trifluoroacetic Acid SCHEMBL3226733 0.65 SSTR4 (0.33)
SCHEMBL24510428 0.65
SCHEMBL24510435 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115003673-A Dihydropyrimidine compound, and preparation method and application thereof 上海维申医药有限公司 2022-09-02 CN disclosed
WO-2022121844-A1 DIHYDROPYRIMIDINE COMPOUND, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 上海维申医药有限公司 2022-06-16 WO disclosed
CN-114621219-A Dihydropyrimidine compound, and preparation method and application thereof 上海维申医药有限公司 2022-06-14 CN disclosed