SCHEMBL24516488

SCHEMBL24516488

COc1ccc(C2C(=O)C=C[C@@H]2O)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 2/20 0.45
EDNRB P24530 1/20 0.45
ALDH1A1 P00352 4/20 0.44
SMN1; SMN2 Q16637 2/20 0.42
MAOA P21397 2/20 0.42
TP53 P04637 2/20 0.42
NPC1 O15118 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
PTGS2 P35354 1/20 0.42
RAB9A P51151 1/20 0.42
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA12 O43570 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
KDM1A O60341 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24516982 0.81 EDNRA (0.42) EDNRAEDNRBALDH1A1SMN1; SMN2MAOA
SCHEMBL24516480 0.80 KDM4E (0.46) ALDH1A1SMN1; SMN2NPC1MAPTHPGD
SCHEMBL24516477 0.78 SLC6A3 (0.40) ALDH1A1SMN1; SMN2HPGDRAB9AKDM4E
SCHEMBL10745108 0.77 EDNRA (0.39) EDNRAEDNRBALDH1A1SMN1; SMN2TP53
SCHEMBL24515872 0.77 EDNRA (0.39) EDNRAEDNRBALDH1A1SMN1; SMN2TP53
SCHEMBL10844446 0.74 ALDH1A1 (0.62) EDNRAEDNRBALDH1A1SMN1; SMN2MAOA
SCHEMBL6758446 0.74 SMN1; SMN2 (0.49) EDNRAEDNRBALDH1A1SMN1; SMN2MAOA
SCHEMBL24516529 0.74 NOS3 (0.37) ALDH1A1NPC1RAB9ACA1CA2
SCHEMBL24516008 0.72 ESR1 (0.43) CES2CES1KDM4E
SCHEMBL24516512 0.72 ALDH1A1 (0.49) EDNRAEDNRBALDH1A1SMN1; SMN2MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022122975-A1 CYCLOPENTENONES DERIVATIVES AND THEIR USE AS ANTIBIOTICS CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2022-06-16 WO disclosed