SCHEMBL24523764

SCHEMBL24523764

N#Cc1cc(-c2ccccc2-c2ccccc2)c2c3cccc4c5c(-c6ccccc6-c6ccccc6)cc(C#N)cc5n(c2c1)c34

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.36
CYP19A1 P11511 1/20 0.36
CYP1A2 P05177 4/20 0.34
MEN1 O00255 4/20 0.34
KMT2A Q03164 4/20 0.34
ALDH1A1 P00352 3/20 0.34
CYP3A4 P08684 3/20 0.34
CLK4 Q9HAZ1 3/20 0.34
HSD17B10 Q99714 3/20 0.34
MAPK1 P28482 2/20 0.34
CYP2C19 P33261 2/20 0.34
LMNA P02545 2/20 0.34
USP2 O75604 2/20 0.34
CYP2D6 P10635 2/20 0.34
ALOX15 P16050 1/20 0.34
HIF1A Q16665 1/20 0.34
KDM4E B2RXH2 2/20 0.33
MAPT P10636 2/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24523908 0.93 METAP2 (0.43) METAP2PTGDR2CYP19A1CYP1A2MEN1
SCHEMBL24523751 0.91 METAP2 (0.39) METAP2PTGDR2CYP19A1CYP1A2MEN1
SCHEMBL24523753 0.90 METAP2 (0.41) METAP2PTGDR2CYP19A1CYP1A2MEN1
SCHEMBL24523739 0.86 METAP2 (0.37) METAP2PTGDR2CYP19A1CYP1A2MEN1
SCHEMBL24524246 0.81 ALDH1A1 (0.35) METAP2PTGDR2CYP19A1CYP1A2MEN1
SCHEMBL24524243 0.81 PRKDC (0.33) CYP1A2ALDH1A1CYP2C19TP53SLC22A12
SCHEMBL24524240 0.77 BRD1 (0.37) ALDH1A1MAPK1LMNAMAPTTDP1
SCHEMBL24523765 0.75 PTGDR2 (0.40) METAP2PTGDR2CYP19A1MEN1KMT2A
SCHEMBL24523768 0.74 MAOA (0.38) CYP19A1CYP1A2ALDH1A1CYP2C19KDM4E
SCHEMBL24524241 0.74 BRD1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129116-A1 INDOLO[3.2.1-JK]CARBAZOLE-6-CARBONITRILE DERIVATIVES AS BLUE FLUORESCENT EMITTERS FOR USE IN OLEDS MERCK PATENT GMBH (DE) 2022-06-23 WO disclosed