SCHEMBL24523786

SCHEMBL24523786

N#Cc1ccc2c3cc(-c4c(-c5ccccc5)nc(-c5ccccc5)nc4-c4ccccc4)cc4c5ccc(C#N)cc5n(c2c1)c34

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 9/20 0.40
ABCB1 P08183 4/20 0.40
HSD17B10 Q99714 2/20 0.39
ADORA2A P29274 2/20 0.39
ADORA1 P30542 2/20 0.39
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2C19 P33261 2/20 0.38
CLK4 Q9HAZ1 2/20 0.38
LMNA P02545 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
ABCC1 P33527 1/20 0.36
ADK P55263 1/20 0.36
MAPK1 P28482 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24523791 0.89 ABCG2 (0.44) ABCG2ABCB1HSD17B10MEN1KMT2A
SCHEMBL24524214 0.88 CYP1A2 (0.35) ABCG2ABCB1HSD17B10ADORA2AMEN1
SCHEMBL24523779 0.84 ABCG2 (0.45) ABCG2ABCB1HSD17B10MEN1KMT2A
SCHEMBL24523727 0.82 CYP1A2 (0.40) ABCG2ABCB1HSD17B10ADORA2AADORA1
SCHEMBL24523719 0.82 MEN1 (0.39) MEN1KMT2A
SCHEMBL24523804 0.81 GABRA1 (0.39) MEN1KMT2A
SCHEMBL24523724 0.81 GABRA1 (0.39) MEN1KMT2A
SCHEMBL24523722 0.81 MEN1 (0.38) MEN1KMT2A
SCHEMBL24523734 0.80 MEN1 (0.40) ADORA2AMEN1KMT2A
SCHEMBL24523765 0.78 PTGDR2 (0.40) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129116-A1 INDOLO[3.2.1-JK]CARBAZOLE-6-CARBONITRILE DERIVATIVES AS BLUE FLUORESCENT EMITTERS FOR USE IN OLEDS MERCK PATENT GMBH (DE) 2022-06-23 WO disclosed