SCHEMBL24526643

SCHEMBL24526643

COCc1cnn(C)c1-c1cc(F)cc(C(=O)OC)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.36
HTR2C P28335 4/20 0.36
POLB P06746 1/20 0.36
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
GRM5 P41594 1/20 0.34
KDM5A P29375 1/20 0.34
KDM5B Q9UGL1 1/20 0.34
OPRL1 P41146 1/20 0.34
MAPT P10636 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
PDE1C Q14123 1/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29759272 1.00 HTR2A (0.36) HTR2AHTR2CPOLBCYP11B1CYP11B2
SCHEMBL24526702 0.90 HTR2A (0.38) HTR2AHTR2CPOLBCYP11B1CYP11B2
SCHEMBL29759212 0.89 HCAR1 (0.38) HTR2AHTR2CKDM5AKDM5BOPRL1
SCHEMBL24526557 0.89 HCAR1 (0.38) HTR2AHTR2CKDM5AKDM5BOPRL1
SCHEMBL6164489 0.82 DGAT2 (0.45) CA12CA1CA2CA9GRM5
SCHEMBL24527049 0.81 HTR2A (0.43) HTR2AHTR2CPOLBCYP11B1CYP11B2
SCHEMBL24526583 0.81 GRIN3B (0.36)
SCHEMBL24526826 0.77 KDM4E (0.38) POLBCYP11B1CYP11B2CA12CA1
SCHEMBL24526566 0.76 ADCY10 (0.39) POLBCYP11B1CYP11B2CA12CA1
SCHEMBL29759314 0.76 ADCY10 (0.39) POLBCYP11B1CYP11B2CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129047-A2 NOVEL MODULATORS OF THE NMDA RECEPTOR H. LUNDBECK A/S (DK) 2022-06-23 WO disclosed