SCHEMBL24528609

SCHEMBL24528609

O=Cc1ccc(-c2nc(-c3ccc(C=O)cc3)c3ncn(-c4ccccc4)c3n2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.44
ADORA2A P29274 1/20 0.43
EGFR P00533 1/20 0.40
PI4KA P42356 1/20 0.40
PI4K2B Q8TCG2 1/20 0.40
PI4K2A Q9BTU6 1/20 0.40
PI4KB Q9UBF8 1/20 0.40
CCNB2 O95067 2/20 0.38
CDK1 P06493 2/20 0.38
CCNB1 P14635 2/20 0.38
CDK5 Q00535 2/20 0.38
CDK5R1 Q15078 2/20 0.38
CCNB3 Q8WWL7 2/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPT P10636 1/20 0.38
PTGS2 P35354 1/20 0.37
FGFR1 P11362 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25733152 0.84 SMN1; SMN2 (0.44) XDHADORA2AEGFRPI4KAPI4K2B
SCHEMBL24528584 0.81 ALDH1A1 (0.37) ALDH1A1MAPTPTGS2POLB
SCHEMBL29681058 0.81 ALDH1A1 (0.37) ALDH1A1MAPTPTGS2POLB
SCHEMBL29681135 0.77 ALDH1A1 (0.39) ALDH1A1MAPTPTGS2
SCHEMBL24528654 0.77 ALDH1A1 (0.39) ALDH1A1MAPTPTGS2
SCHEMBL24528639 0.76 ATM (0.37) XDHADORA2AALDH1A1FGFR1
SCHEMBL24528680 0.75 ALDH1A1 (0.40) ALDH1A1MAPTPTGS2
SCHEMBL29680897 0.74 PIK3CA (0.46) ALDH1A1MAPTTSHRPOLB
SCHEMBL29681271 0.73 ALDH1A1 (0.39) CCNB2CDK1CCNB1CDK5CDK5R1
SCHEMBL24528681 0.73 ALDH1A1 (0.39) CCNB2CDK1CCNB1CDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed