SCHEMBL25733152

SCHEMBL25733152

c1ccc(-n2cnc3c(-c4ccncc4)nc(-c4ccncc4)nc32)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.44
ADORA2A P29274 1/20 0.44
XDH P47989 1/20 0.43
KMT2A Q03164 4/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP1A2 P05177 1/20 0.41
POLB P06746 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.41
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
EGFR P00533 1/20 0.41
PI4KA P42356 1/20 0.41
PI4K2B Q8TCG2 1/20 0.41
PI4K2A Q9BTU6 1/20 0.41
PI4KB Q9UBF8 1/20 0.41
DYRK1A Q13627 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26315304 0.85 CYP2D6 (0.50) SMN1; SMN2ADORA2AXDHKMT2ACYP2D6
SCHEMBL24528609 0.84 XDH (0.44) ADORA2AXDHCYP2D6CYP2C9CYP2C19
SCHEMBL25618869 0.77 PIK3CA (0.48) CYP2C9CYP2C19CYP1A2CYP3A4MAPT
SCHEMBL28143395 0.72 DPP4 (0.41) ADORA2AKMT2APOLBHTTMEN1
SCHEMBL28295500 0.72 MAPK14 (0.49) ADORA2AKMT2AMAPTHTTMEN1
SCHEMBL28143391 0.70 ADORA2A (0.60) SMN1; SMN2ADORA2AXDHKMT2AEGFR
SCHEMBL28143392 0.70 ADORA2A (0.60) ADORA2AXDHCYP2D6CYP1A2POLB
SCHEMBL24500181 0.68 ALDH1A1 (0.52) SMN1; SMN2ADORA2AKMT2AMAPTHTT
SCHEMBL30560080 0.68 ALDH1A1 (0.52) SMN1; SMN2ADORA2AKMT2AMAPTHTT
SCHEMBL300860 0.67 KDM4E (0.46) XDHPI4KAPI4K2BPI4K2API4KB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119031913-A Purine and methods of use thereof 奇尼塔公司 2024-11-26 CN disclosed
CN-118946360-A Bicyclic heteroarenes and methods of use thereof 奇尼塔公司 2024-11-12 CN disclosed
EP-4444312-A2 PURINES AND METHODS OF THEIR USE Kineta, Inc. (US) 2024-10-16 EP disclosed
WO-2023107552-A2 PURINES AND METHODS OF THEIR USE Kineta, Inc. (US) 2023-06-15 WO disclosed
WO-2023107552-A2 PURINES AND METHODS OF THEIR USE Kineta, Inc. (US) 2023-06-15 WO disclosed
EP-4161519-A1 PURINES AND METHODS OF THEIR USE Yumanity Therapeutics, Inc. (US) 2023-04-12 EP disclosed