SCHEMBL24528670

SCHEMBL24528670

CNCc1c(Nc2ccccc2)nc(-c2ccc(/C=N/CCCCCN(C)C)cc2)nc1-c1ccc(/C=N\CCCCCN(C)C)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAD52 P43351 3/20 0.35
MAPK1 P28482 3/20 0.35
ALDH1A1 P00352 2/20 0.35
POLB P06746 3/20 0.35
USP2 O75604 2/20 0.34
LMNA P02545 2/20 0.34
TP53 P04637 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
TSHR P16473 2/20 0.34
CYP2C19 P33261 2/20 0.34
CLK4 Q9HAZ1 1/20 0.34
ESR1 P03372 1/20 0.34
RXFP1 Q9HBX9 1/20 0.33
TLR9 Q9NR96 1/20 0.33
KDM1A O60341 5/20 0.33
MEN1 O00255 2/20 0.33
MAPT P10636 2/20 0.33
KMT2A Q03164 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24528616 0.99 RAD52 (0.36) RAD52MAPK1ALDH1A1POLBUSP2
SCHEMBL24528631 0.96 RAD52 (0.36) RAD52MAPK1ALDH1A1POLBUSP2
SCHEMBL24528607 0.82 TLR9 (0.36) MAPK1ALDH1A1POLBTLR9MAPT
SCHEMBL24528713 0.77 PDE4B (0.41) MAPK1ALDH1A1POLBUSP2LMNA
SCHEMBL24528677 0.73 KDM4E (0.34) RAD52MAPK1ALDH1A1POLBLMNA
SCHEMBL24528599 0.73 KDM4E (0.33) RAD52MAPK1ALDH1A1POLBLMNA
SCHEMBL24528695 0.72 KDM4E (0.34) RAD52MAPK1ALDH1A1POLBLMNA
SCHEMBL24528655 0.72 KDM4E (0.34) RAD52MAPK1ALDH1A1POLBLMNA
SCHEMBL24528691 0.72 PDE5A (0.35) RAD52RXRANR4A2
SCHEMBL24528668 0.71 RAD52 (0.32) RAD52ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed