SCHEMBL24528607

SCHEMBL24528607

CNCc1c(Nc2ccccc2)nc(-c2ccc(/C=N/CCCCN3CCN(C)CC3)cc2)nc1-c1ccc(/C=N\CCCCN2CCN(C)CC2)cc1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 4/20 0.36
HRH4 Q9H3N8 1/20 0.36
CFTR P13569 1/20 0.35
KDM4E B2RXH2 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
RAB9A P51151 2/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
NPC1 O15118 1/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
FLT3 P36888 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24528616 0.83 RAD52 (0.36) TLR9KDM4ESMN1; SMN2ALDH1A1POLB
SCHEMBL24528670 0.82 RAD52 (0.35) TLR9KDM4ESMN1; SMN2ALDH1A1POLB
SCHEMBL24528631 0.82 RAD52 (0.36) TLR9KDM4ESMN1; SMN2ALDH1A1POLB
SCHEMBL24528661 0.76 RAD52 (0.36) TLR9KDM4ESMN1; SMN2RAB9AALDH1A1
SCHEMBL24528713 0.74 PDE4B (0.41) KDM4ESMN1; SMN2ALDH1A1POLBMAPT
SCHEMBL24528690 0.74 TLR9 (0.41) TLR9KDM4ESMN1; SMN2RAB9AALDH1A1
SCHEMBL29680767 0.73 KDM5B (0.42) KDM4EALDH1A1MAPTMAPK1
SCHEMBL24528686 0.73 RAB9A (0.35) TLR9KDM4ESMN1; SMN2RAB9AALDH1A1
SCHEMBL24528648 0.73 RAD52 (0.37) TLR9KDM4ESMN1; SMN2RAB9AALDH1A1
SCHEMBL29680554 0.73 RAD52 (0.37) TLR9KDM4ESMN1; SMN2RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed