SCHEMBL2453347

SCHEMBL2453347

CC(=O)c1ccc(Oc2ncnc(N)c2C=O)cc1C

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.46
KDR P35968 17/20 0.43
RET P07949 4/20 0.43
CSF1R P07333 1/20 0.40
KIT P10721 1/20 0.40
PDGFRA P16234 1/20 0.40
FLT1 P17948 1/20 0.40
FLT4 P35916 1/20 0.40
FLT3 P36888 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2450805 0.85 RET (0.64) KDRRETCSF1RKITPDGFRA
SCHEMBL5322205 0.85 RET (0.47) ALDH1A1KDRRETCSF1RKIT
SCHEMBL5322198 0.85 RET (0.47) ALDH1A1KDRRETCSF1RKIT
SCHEMBL2450807 0.85 RET (0.64) KDRRETCSF1RKITPDGFRA
SCHEMBL2448477 0.75 RET (0.65) KDRRETCSF1RKITPDGFRA
SCHEMBL2450638 0.75 RET (0.54) ALDH1A1KDRRETPDGFRA
SCHEMBL2454635 0.74 KDR (0.74) ALDH1A1KDRRET
SCHEMBL2453476 0.74 RET (0.45) KDRRET
SCHEMBL2451070 0.74 RET (0.48) KDRRETCSF1RKITPDGFRA
SCHEMBL2450822 0.73 RET (0.62) KDRRETCSF1RKITPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007109783-A2 SUBSTITUTED PYRIMIDINE KINASE INHIBITORS JANSSEN PHARMACEUTICA, N.V. (BE) 2007-09-27 WO claimed
US-8013153-B2 Substituted pyrimidine kinase inhibitors JANSSEN PHARMACEUTICA, N.V. (BE) 2011-09-06 US disclosed
US-20070254896-A1 SUBSTITUTED PYRIMIDINE KINASE INHIBITORS JANSSEN PHARMACEUTICA, N.V. (BE) 2007-11-01 US disclosed
WO-2007109783-A2 SUBSTITUTED PYRIMIDINE KINASE INHIBITORS JANSSEN PHARMACEUTICA, N.V. (BE) 2007-09-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070254896-A1 SUBSTITUTED PYRIMIDINE KINASE INHIBITORS DTYMK, TK1, DCK ALDH1A1 2496/4885KDR 1975/4885RET 577/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.