SCHEMBL24533960

SCHEMBL24533960

CCC(F)(F)c1cncc(Br)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
POLB P06746 1/20 0.37
HCAR2 Q8TDS4 1/20 0.37
KDM4E B2RXH2 1/20 0.37
HTT P42858 3/20 0.36
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
RAB9A P51151 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
PRKAB2 O43741 1/20 0.34
PRKAG1 P54619 1/20 0.34
PRKAA2 P54646 1/20 0.34
PRKAA1 Q13131 1/20 0.34
PRKAG3 Q9UGI9 1/20 0.34
PRKAG2 Q9UGJ0 1/20 0.34
PRKAB1 Q9Y478 1/20 0.34
SLC22A12 Q96S37 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22004473 0.78 POLB (0.38) CYP11B1CYP11B2POLBHCAR2KDM4E
SCHEMBL3507833 0.78 CYP11B1 (0.42) CYP11B1CYP11B2POLBHCAR2KDM4E
SCHEMBL24534060 0.78 CYP11B1 (0.42) CYP11B1CYP11B2POLBHCAR2KDM4E
SCHEMBL185547 0.77 CYP11B1 (0.49) CYP11B1CYP11B2POLBHCAR2CYP3A4
SCHEMBL29920114 0.77 CYP11B1 (0.49) CYP11B1CYP11B2POLBHCAR2CYP3A4
SCHEMBL22658213 0.77 KDM4E (0.33) KDM4E
SCHEMBL25480051 0.74 CYP11B1 (0.41) CYP11B1CYP11B2CYP1A2CYP3A4SLC22A12
SCHEMBL2732538 0.73 CYP1A2 (0.39) CYP11B1CYP11B2POLBHCAR2KDM4E
SCHEMBL433999 0.72 CYP11B2 (0.44) CYP11B1CYP11B2
SCHEMBL16751902 0.71 POLB (0.44) POLBHCAR2KDM4EHTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022128850-A1 NOVEL ISOQUINOLINE DERIVATIVES AND PHARMACEUTICAL COPOSITIONS THEREOF FOR THE TREATMENT OF DISEASES GALAPAGOS NV (BE) 2022-06-23 WO disclosed