SCHEMBL24534129

SCHEMBL24534129

FC(F)C1(c2cncc(N=C(c3ccccc3)c3ccccc3)c2)CC1

nearest known ligand 0.34

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
OPRD1 P41143 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31058636 0.81 ESR2 (0.42) ESR1ESR2OPRD1
SCHEMBL24534130 0.77 ALDH1A1 (0.37) ESR1ESR2OPRD1
SCHEMBL30042841 0.76 ESR1 (0.39) ESR1ESR2
SCHEMBL23540686 0.76 ESR1 (0.39) ESR1ESR2
SCHEMBL23540714 0.74 ESR1 (0.38) ESR1ESR2
SCHEMBL30015180 0.74 ESR1 (0.38) ESR1ESR2
SCHEMBL29112221 0.70 ESR1 (0.46) ESR1ESR2
SCHEMBL15542419 0.70 ESR1 (0.50) ESR1ESR2
SCHEMBL31226463 0.69 AKT1 (0.40)
SCHEMBL15542113 0.68 ESR1 (0.41) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022128850-A1 NOVEL ISOQUINOLINE DERIVATIVES AND PHARMACEUTICAL COPOSITIONS THEREOF FOR THE TREATMENT OF DISEASES GALAPAGOS NV (BE) 2022-06-23 WO disclosed