SCHEMBL2453480

SCHEMBL2453480

CCc1[nH]c2ncnn2c(=O)c1Cc1ccc(Cl)c(C(F)(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MBOAT4 Q96T53 5/20 0.39
KDM4A O75164 1/20 0.39
KDM5A P29375 1/20 0.39
KDM5B Q9UGL1 1/20 0.39
ADORA2B P29275 1/20 0.38
PDE2A O00408 1/20 0.37
MAOB P27338 2/20 0.37
PLA2G7 Q13093 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
NR3C1 P04150 1/20 0.35
P2RX7 Q99572 2/20 0.35
IDO1 P14902 1/20 0.34
AR P10275 1/20 0.34
COMT P21964 1/20 0.34
KCNN4 O15554 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2455141 0.88 KDM4A (0.39) MBOAT4KDM4AKDM5AKDM5BPDE2A
SCHEMBL2464506 0.88 MBOAT4 (0.40) MBOAT4KDM4AKDM5AKDM5BADORA2B
SCHEMBL2465551 0.88 MBOAT4 (0.40) MBOAT4KDM4AKDM5AKDM5BADORA2B
SCHEMBL2466816 0.87 ALKBH3 (0.39) MAOB
SCHEMBL2456758 0.82 KDM4A (0.38) MBOAT4KDM4AKDM5AKDM5BADORA2B
SCHEMBL2456756 0.81 PDE2A (0.46) MBOAT4KDM4AKDM5AKDM5BPDE2A
SCHEMBL2456189 0.77 NR3C2 (0.37) MBOAT4ADORA2BPDE2AP2RX7AR
SCHEMBL2541935 0.77 MBOAT4 (0.37) MBOAT4ADORA2BPDE2AP2RX7AR
SCHEMBL2457055 0.71 AR (0.35) MBOAT4ADORA2BPDE2AP2RX7AR
SCHEMBL12324705 0.71 KDM4A (0.36) KDM4AKDM5AKDM5BMAOBP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011114148-A1 4H- [1, 2, 4] TRIAZOLO [5, 1 -B] PYRIMIDIN-7 -ONE DERIVATIVES AS CCR2B RECEPTOR ANTAGONISTS ASTRAZENECA AB (SE) 2011-09-22 WO claimed
WO-2011114148-A1 4H- [1, 2, 4] TRIAZOLO [5, 1 -B] PYRIMIDIN-7 -ONE DERIVATIVES AS CCR2B RECEPTOR ANTAGONISTS ASTRAZENECA AB (SE) 2011-09-22 WO disclosed