SCHEMBL2454487

SCHEMBL2454487

CCNS(=O)(=O)N(CC)c1ccc2ccc3ncc(-c4cnn(C)c4)cc3c(=O)c2c1

nearest known ligand 0.67

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MET P08581 20/20 0.67
MST1R Q04912 1/20 0.62
KCNH2 Q12809 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2446196 0.90 MET (0.76) METMST1RKCNH2
SCHEMBL2322770 0.81 MET (0.72) METMST1RKCNH2
SCHEMBL2446680 0.80 MET (0.67) METMST1RKCNH2
SCHEMBL2443744 0.80 MET (1.00) METMST1RKCNH2
SCHEMBL2447126 0.80 MET (0.64) METMST1RKCNH2
SCHEMBL2452747 0.79 MET (0.69) METMST1RKCNH2
SCHEMBL2447035 0.79 MET (0.81) METMST1R
SCHEMBL2446421 0.79 MET (0.85) METMST1RKCNH2
SCHEMBL3952870 0.79 MET (0.69) METMST1RKCNH2
SCHEMBL3948881 0.79 MET (0.58) METMST1RKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1896421-B1 BENZOCYCLOHEPTAPYRIDINES AS INHIBITORS OF THE RECEPTOR TYROSINE KINASE MET MERCK SHARP & DOHME (US) 2011-09-14 EP claimed
EP-1896421-B1 BENZOCYCLOHEPTAPYRIDINES AS INHIBITORS OF THE RECEPTOR TYROSINE KINASE MET MERCK SHARP & DOHME (US) 2011-09-14 EP disclosed